mTOR Inhibitors

Name
mTOR Inhibitors
Accession Number
DBCAT004158
Description

Medications that exert their immunosuppressive effects via inhibition of the mammalian target of rapamycin (mTOR)

Drugs
DrugDrug Description
AZD-8055AZD8055 has been used in trials studying the treatment of Cancer, Lymphomas, Solid Tumors, MALIGNANT GLIOMA, and brainstem glioma, among others.
EverolimusA mammalian target of rapamycin (mTOR) kinase inhibitor used to treat various types of malignancies.
GedatolisibA pan-PI3K and mTORC1/2 inhibitor used as part of a second-line chemotherapy regimen for HR-positive, HER2-negative advanced breast cancer without a PIK3CA mutation following endocrine therapy.
GSK-1059615GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.
OSI-027OSI-027 has been used in trials studying the treatment of Any Solid Tumor or Lymphoma.
PimecrolimusA topical calcineurin inhibitor used in the treatment of mild-moderate atopic dermatitis who are not candidates for other types of therapy due to previous lack of response or other reasons.
RidaforolimusInvestigated for use/treatment in solid tumors, sarcoma, cancer/tumors (unspecified), endometrial cancer, prostate cancer, and bone metastases.
SirolimusAn mTOR inhibitor immunosuppressant used to prevent organ transplant rejections, treat lymphangioleiomyomatosis, and treat adults with perivascular epithelioid cell tumors.
TemsirolimusA antineoplastic agent used in the treatment of renal cell carcinoma (RCC) that works by inhibiting mTOR.
VistusertibVistusertib is under investigation for the treatment of Advanced Gastric Adenocarcinoma.
Drugs & Drug Targets
DrugTargetType
AZD-8055Serine/threonine-protein kinase mTORtarget
EverolimusSerine/threonine-protein kinase mTORtarget
EverolimusCytochrome P450 3A4enzyme
EverolimusSolute carrier organic anion transporter family member 1B1transporter
EverolimusSolute carrier organic anion transporter family member 1B3transporter
EverolimusSolute carrier organic anion transporter family member 1A2transporter
EverolimusCytochrome P450 2D6enzyme
EverolimusATP-dependent translocase ABCB1transporter
EverolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
GedatolisibPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformtarget
GedatolisibSerine/threonine-protein kinase mTORtarget
GSK-1059615Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoformtarget
GSK-1059615Phosphatidylinositol 3-kinase catalytic subunit type 3target
GSK-1059615Serine/threonine-protein kinase mTORtarget
OSI-027Serine/threonine-protein kinase mTORtarget
PimecrolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
PimecrolimusSerine/threonine-protein kinase mTORtarget
PimecrolimusCytochrome P450 3A4enzyme
PimecrolimusProtein phosphatase 3 catalytic subunit alphatarget
RidaforolimusSerine/threonine-protein kinase mTORtarget
RidaforolimusCytochrome P450 3A4enzyme
SirolimusCytochrome P450 3A5enzyme
SirolimusCytochrome P450 3A7enzyme
SirolimusATP-dependent translocase ABCB1transporter
SirolimusSolute carrier organic anion transporter family member 1B1transporter
SirolimusMultidrug and toxin extrusion protein 1transporter
SirolimusAlbumincarrier
SirolimusAlpha-1-acid glycoprotein 1carrier
SirolimusApolipoproteinscarrier
SirolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
SirolimusSerine/threonine-protein kinase mTORtarget
SirolimusCytochrome P450 3A4enzyme
TemsirolimusPeptidyl-prolyl cis-trans isomerase FKBP1Atarget
TemsirolimusATP-dependent translocase ABCB1transporter
TemsirolimusCytochrome P450 2D6enzyme
TemsirolimusCytochrome P450 3A7enzyme
TemsirolimusCytochrome P450 3A5enzyme
TemsirolimusSerine/threonine-protein kinase mTORtarget
TemsirolimusCytochrome P450 3A4enzyme
VistusertibSerine/threonine-protein kinase mTORtarget
VistusertibTarget of rapamycin complex 2 subunit MAPKAP1target