Bile Salt Export Pump Inhibitors

Name
Bile Salt Export Pump Inhibitors
Accession Number
DBCAT005493
Description

Not Available

Drugs
DrugDrug Description
AvapritinibA selective tyrosine kinase inhibitor being investigated for the treatment of multidrug resistant gastrointestinal tumors.
RomidepsinA histone deacetylase (HDAC) inhibitor used to treat cutaneous T-cell lymphoma.
Drugs & Drug Targets
DrugTargetType
AvapritinibPlatelet derived growth factor receptor alphatarget
AvapritinibMast/stem cell growth factor receptor Kittarget
AvapritinibP-glycoprotein 1transporter
AvapritinibATP-binding cassette sub-family G member 2transporter
AvapritinibCytochrome P450 3A4enzyme
AvapritinibCytochrome P450 2C9enzyme
AvapritinibBile salt export pumptransporter
AvapritinibMultidrug and toxin extrusion protein 1transporter
AvapritinibMultidrug and toxin extrusion protein 2transporter
RomidepsinCytochrome P450 3A4enzyme
RomidepsinCytochrome P450 3A5enzyme
RomidepsinP-glycoprotein 1transporter
RomidepsinSolute carrier organic anion transporter family member 1B3transporter
RomidepsinCytochrome P450 1A1enzyme
RomidepsinCytochrome P450 2B6enzyme
RomidepsinCytochrome P450 2C19enzyme
RomidepsinHistone deacetylase 1target
RomidepsinHistone deacetylase 2target
RomidepsinHistone deacetylase 4target
RomidepsinHistone deacetylase 6target
RomidepsinMultidrug resistance-associated protein 1target
RomidepsinBile salt export pumptransporter
RomidepsinSolute carrier organic anion transporter family member 1B1transporter
RomidepsinSolute carrier family 22 member 6transporter
RomidepsinSolute carrier family 22 member 2transporter
RomidepsinHistone deacetylasetarget