Selective Estrogen Receptor Degraders

Name
Selective Estrogen Receptor Degraders
Accession Number
DBCAT005805
Description

Not Available

Drugs
DrugDrug Description
ElacestrantAn estrogen receptor antagonist used to treat ER-positive, HER2-negative, ESR1-mutated advanced or metastatic breast cancer with disease progression following at least one line of endocrine therapy.
Drugs & Drug Targets
DrugTargetType
ElacestrantEstrogen receptor alphatarget
ElacestrantCytochrome P450 3A4enzyme
ElacestrantCytochrome P450 2A6enzyme
ElacestrantCytochrome P450 2C9enzyme
ElacestrantSolute carrier organic anion transporter family member 2B1transporter
ElacestrantP-glycoprotein 1transporter
ElacestrantATP-binding cassette sub-family G member 2transporter