Adrenergic beta-Agonists

Name
Adrenergic beta-Agonists
Accession Number
DBCAT000553
Description

Drugs that selectively bind to and activate beta-adrenergic receptors.

Drugs
DrugDrug Description
AbediterolAbediterol has been used in trials studying the treatment of Asthma, Chronic Obstructive Pulmonary Disease (COPD), and Chronic Obstructive Pulmonary Disease (COPD) and Asthma.
AlbuterolA beta-2 adrenergic receptor agonist used to treat asthma, bronchitis, COPD, as well as prevent exercise induced bronchospasms.
AmibegronInvestigated for use/treatment in depression, irritable bowel syndrome (IBS), and obesity.
ArbutamineUsed to elicit acute cardiovascular responses (cardiac stumulant), similar to those produced by exercise, in order to aid in diagnosing the presence or absence of coronary artery disease (CAD) in...
ArformoterolA beta-2 adrenergic agonist and bronchodilator used for long-term, symptomatic treatment of reversible bronchoconstriction in patients with chronic obstructive pulmonary disease (COPD), including chronic bronchitis and emphysema.
BambuterolA long acting beta2-adrenoceptor agonist for the management of lung diseases associated with bronchospasm.
BatefenterolBatefenterol has been used in trials studying the treatment of Pulmonary Disease, Chronic Obstructive.
BefunololUsed in the management of open angle glaucoma. PMID: 12480285.
BitolterolUsed to dilate air passages in the lungs that have become narrowed as a result of disease or inflammation. It is used in the treatment of asthma and chronic obstructive...
CeliprololA beta-blocker for the management of hypertension and angina pectoris.
ClenbuterolA decongestant and bronchodilator used in a variety of respiratory conditions.
DenopamineDenopamine is a small molecule drug. Denopamine has a monoisotopic molecular weight of 317.16 Da.
DipivefrinA prodrug of epinephrine used in ophthalmic solutions to reduce intraocular pressure in chronic open-angle glaucoma.
DobutamineA beta-1 agonist used to treat cardiac decompensation in patients with organic heart disease or from cardiac surgery.
DopexamineDopexamine has been used in trials studying the diagnostic and treatment of Free Flap, Oral Cancer, Hypotension, Septic Shock, and Head and Neck Cancer.
DoxofyllineA methylxanthine derivative used in chronic obstructive pulmonary disease, asthma, and bronchospasms.
DroxidopaA medication used to treat symptomatic neurogenic orthostatic hypotension (nOH) caused by dopamine beta-hydroxylase deficiency, non-diabetic autonomic neuropathy and primary autonomic failure caused by conditions such as Parkinson's disease.
Ephedra sinica rootAn alpha and beta-adrenergic agonist used for the management of respiratory conditions related to bronchial asthma, such as wheezing, shortness of breath, and tightness of chest.
EphedrineAn alpha and beta-adrenergic agonist indicated to treat hypotension under anesthesia, allergic conditions, bronchial asthma, and nasal congestion.
EpinephrineA hormone and neurotransmitter used to treat allergic reactions, to restore cardiac rhythm, and to control mucosal congestion, glaucoma, and asthma.
EtafedrineA beta-2 adrenoceptor agonist used to treat a cough associated with inflamed mucosa.
EtilefrineAn adrenergic agonist primarily of α1 and β1 receptors used as an anti-hypotensive.
FenoterolA beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
FormoterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
HexoprenalineHexoprenaline is a stimulant of beta 2 adrenergic receptors. It is used as a bronchodilator, antiasthmatic, and tocolytic agent.
HigenamineHigenamine is under investigation in clinical trial NCT01451229 (Pharmacokinetics and Pharmacodynamics of Higenamine in Chinese Healthy Subjects).
IndacaterolAn inhaled long-acting beta-2 adrenergic agonist used to relax bronchial smooth muscle and improve symptoms and airflow obstruction caused by Chronic Obstructive Pulmonary Disease (COPD) and moderate to severe asthma.
IsoetharineFor the treatment of asthma, wheezing, and chronic asthmatic bronchitis.
IsoprenalineA catecholamine non-selective beta-adrenergic agonist typically used to treat bradycardia and heart block.
IsoxsuprineA beta-adrenergic agonist used in the symptomatic treatment of cerebrovascular insufficiency, peripheral vascular disease of arteriosclerosis obliterans, thromboangiitis obliterans (Buerger's disease) and Raynaud's disease.
LAS-190792Not Annotated
LevosalbutamolA beta-2 adrenergic receptor agonist used to treat COPD and asthma.
LidamidineLidamidine is a small molecule drug. Lidamidine has a monoisotopic molecular weight of 220.13 Da.
MethoxyphenamineNot Annotated
MirabegronA beta-3 adrenergic agonist used to treat overactive bladder and neurogenic detrusor overactivity.
NebivololA beta blocking agent used to treat hypertension and aid in the management of heart failure.
NorepinephrineA sympathomimetic used in the control of blood pressure during various hypotensive states and as an adjunct treatment during cardiac arrest.
NylidrinA vasodilator used to treat patients with peripheral vascular disorders, and elderly patients with symptoms associated with organic mental disorders.
OlodaterolA long-acting beta2-adrenergic agonist used in the management of chronic obstructive pulmonary disease (COPD), including chronic bronchitis and/or emphysema.
OrciprenalineA beta-2 adrenergic agonist used to treat bronchospasm, asthma, and COPD.
OxyfedrineNot Annotated
PF-00610355PF-00610355 has been used in trials studying the treatment of Lung Disease, Moxifloxacin, Pulmonary Disease, Asthma, Bronchial, and Bronchial Diseases, among others.
PhenylpropanolamineA sympathomimetic that was previously used in nasal decongestants and weight loss products, but has been withdrawn by the FDA due to safety risks and lack of efficacy.
PirbuterolA beta-2 adrenergic agonist and bronchodilator used for the symptomatic treatment of asthma.
PrenalterolNot Annotated
ProcaterolA beta-2 adrenergic receptor agonist and bronchodilator used for the treatment of asthma and chronic obstructive pulmonary disease (COPD).
ProtokylolProtokylol is a β-adrenergic receptor agonist used as a bronchodilator in Europe and the United States.
PseudoephedrineAn alpha and beta adrenergic agonist used to treat nasal and sinus congestion, as well as allergic rhinitis.
RacephedrineNot Annotated
RacepinephrineA bronchodilator used to treat intermittent asthma.
RactopamineNot Annotated
ReproterolA short-acting β2 adrenoreceptor agonist used to treat various types of asthma including allergic asthma, non-allergic asthma, and exercise-induced asthma.
RimiterolNot Annotated
RitobegronRitobegron is under investigation in clinical trial NCT02256735 (Study to Investigate the Effect of KUC 7483 CL on the QT/QTc Interval of the ECG in Comparison to Placebo and Moxifloxacin...
RitodrineAn adrenergic beta agonist used to treat premature labor.
SalmeterolA long-acting beta-2 adrenergic receptor agonist used to treat asthma and COPD.
SolabegronInvestigated for use/treatment in diabetes mellitus type 2, irritable bowel syndrome (IBS), and urinary incontinence.
TerbutalineA beta-2 adrenergic agonist used as a bronchodilator and to prevent premature labor.
TretoquinolNot Annotated
TulobuterolAn inhaled long-acting beta2-adrenergic receptor agonist used as a bronchodilator in the management of asthma and COPD.
VibegronA beta-3 adrenergic agonist the treatment of overactive bladder (OAB) with symptoms of urge urinary incontinence, urgency, and urinary frequency in adults.
VilanterolA long-acting beta2-adrenergic agonist used in combination with other bronchodilators for the management of chronic obstructive pulmonary disease (COPD), including chronic bronchitis and/or emphysema.
XamoterolXamoterol is a β1-adrenoceptor partial agonist that has shown to improve systolic and diastolic function in studies with heart failure patients. It modulates the sympathetic control of the heart but...
Drugs & Drug Targets
DrugTargetType
AbediterolBeta-2 adrenergic receptortarget
AlbuterolBeta-2 adrenergic receptortarget
AlbuterolBeta-1 adrenergic receptortarget
AlbuterolCytochrome P450 3A4enzyme
AlbuterolBeta-3 adrenergic receptortarget
AmibegronBeta-3 adrenergic receptortarget
ArbutamineBeta-1 adrenergic receptortarget
ArbutamineBeta-2 adrenergic receptortarget
ArbutamineBeta-3 adrenergic receptortarget
ArformoterolBeta-2 adrenergic receptortarget
ArformoterolAdenylate cyclasetarget
ArformoterolCytochrome P450 2C9enzyme
ArformoterolCytochrome P450 2D6enzyme
ArformoterolCytochrome P450 2C19enzyme
ArformoterolCytochrome P450 2A6enzyme
BambuterolCholinesterasetarget
BambuterolCholinesteraseenzyme
BambuterolBeta-2 adrenergic receptortarget
BatefenterolMuscarinic acetylcholine receptor M3target
BatefenterolMuscarinic acetylcholine receptor M2target
BatefenterolBeta-2 adrenergic receptortarget
BefunololCytochrome P450 2D6enzyme
BefunololBeta-2 adrenergic receptortarget
BefunololBeta-1 adrenergic receptortarget
BitolterolBeta-2 adrenergic receptortarget
BitolterolBeta-3 adrenergic receptortarget
CeliprololBeta-1 adrenergic receptortarget
CeliprololAlpha-2 adrenergic receptorstarget
CeliprololCytochrome P450 2D6enzyme
CeliprololAlpha-2C adrenergic receptortarget
CeliprololAlpha-2B adrenergic receptortarget
CeliprololAlpha-2A adrenergic receptortarget
CeliprololBeta-3 adrenergic receptortarget
CeliprololBeta-2 adrenergic receptortarget
ClenbuterolBeta-2 adrenergic receptortarget
ClenbuterolBeta-nerve growth factortarget
ClenbuterolTumor necrosis factortarget
ClenbuterolBeta-1 adrenergic receptortarget
ClenbuterolBeta-3 adrenergic receptortarget
ClenbuterolCytochrome P450 1A1enzyme
DenopamineD(2) dopamine receptortarget
DipivefrinAlpha-1A adrenergic receptortarget
DipivefrinBeta-1 adrenergic receptortarget
DipivefrinAcetylcholinesterasetarget
DipivefrinBeta-2 adrenergic receptortarget
DipivefrinCholinesterasetarget
DipivefrinAlpha-2A adrenergic receptortarget
DobutamineEstrogen receptortarget
DobutamineBeta-2 adrenergic receptortarget
DobutamineAlpha-1 adrenergic receptorstarget
DobutamineBeta-1 adrenergic receptortarget
DobutamineCatechol O-methyltransferaseenzyme
DopexamineD(2) dopamine receptortarget
DoxofyllineAdenosine receptor A2atarget
DoxofyllineBeta-2 adrenergic receptortarget
DoxofyllineCytochrome P450 1A2enzyme
DoxofyllinecGMP-dependent 3',5'-cyclic phosphodiesterasetarget
DroxidopaSodium-dependent noradrenaline transportertransporter
DroxidopaMonocarboxylate transporter 10transporter
DroxidopaAromatic-L-amino-acid decarboxylaseenzyme
DroxidopaBeta-3 adrenergic receptortarget
DroxidopaBeta-2 adrenergic receptortarget
DroxidopaBeta-1 adrenergic receptortarget
DroxidopaPhenylalanine-4-hydroxylasetarget
DroxidopaAlpha-1A adrenergic receptortarget
DroxidopaAlpha-1B adrenergic receptortarget
DroxidopaAlpha-1D adrenergic receptortarget
DroxidopaAlpha-2A adrenergic receptortarget
DroxidopaAlpha-2B adrenergic receptortarget
DroxidopaAlpha-2C adrenergic receptortarget
Ephedra sinica rootAlpha-2A adrenergic receptortarget
Ephedra sinica rootSodium-dependent dopamine transportertarget
Ephedra sinica rootSynaptic vesicular amine transportertarget
Ephedra sinica rootChromaffin granule amine transportertarget
Ephedra sinica rootSodium-dependent noradrenaline transportertarget
Ephedra sinica rootAmine oxidase [flavin-containing] Atarget
Ephedra sinica rootAmine oxidase [flavin-containing] Btarget
Ephedra sinica rootSodium-dependent serotonin transportertarget
Ephedra sinica rootAlpha-2B adrenergic receptortarget
Ephedra sinica rootAlpha-2C adrenergic receptortarget
Ephedra sinica rootBeta-1 adrenergic receptortarget
Ephedra sinica rootBeta-2 adrenergic receptortarget
Ephedra sinica rootBeta-3 adrenergic receptortarget
EphedrineSynaptic vesicular amine transportertransporter
EphedrineAcetylcholinesteraseenzyme
EphedrineD(2) dopamine receptortarget
EphedrineBeta-2 adrenergic receptortarget
EphedrineBeta-1 adrenergic receptortarget
EphedrineAlbumincarrier
EphedrineCholinesteraseenzyme
EphedrineSodium-dependent noradrenaline transportertarget
EphedrineAlpha-1A adrenergic receptortarget
EpinephrineAlpha-1A adrenergic receptortarget
EpinephrineCatechol O-methyltransferaseenzyme
EpinephrineAlpha-1B adrenergic receptortarget
EpinephrineMonoamine oxidaseenzyme
EpinephrineBeta-1 adrenergic receptortarget
EpinephrineCytochrome P450 2C9enzyme
EpinephrineCytochrome P450 3A4enzyme
EpinephrineAlpha-1D adrenergic receptortarget
EpinephrineBeta-2 adrenergic receptortarget
EpinephrineSolute carrier family 22 member 2transporter
EpinephrineSolute carrier family 22 member 1transporter
EpinephrineTumor necrosis factortarget
EpinephrineAlpha-2B adrenergic receptortarget
EpinephrineAlpha-2A adrenergic receptortarget
EtafedrineBeta-2 adrenergic receptortarget
EtilefrineSolute carrier family 22 member 3transporter
EtilefrineAlpha-1D adrenergic receptortarget
EtilefrineAlpha adrenergic receptortarget
FenoterolBeta-2 adrenergic receptortarget
FenoterolBeta-1 adrenergic receptortarget
FenoterolBeta-3 adrenergic receptortarget
FormoterolSolute carrier family 22 member 3transporter
FormoterolUDP-glucuronosyltransferase 2B7enzyme
FormoterolUDP-glucuronosyltransferase 1A1enzyme
FormoterolBeta-2 adrenergic receptortarget
FormoterolBeta-1 adrenergic receptortarget
FormoterolBeta-3 adrenergic receptortarget
FormoterolCytochrome P450 2D6enzyme
FormoterolCytochrome P450 2C19enzyme
FormoterolCytochrome P450 2C9enzyme
FormoterolCytochrome P450 2A6enzyme
FormoterolUDP-glucuronosyltransferase 1A8enzyme
FormoterolUDP-glucuronosyltransferase 1A9enzyme
FormoterolAlbumincarrier
FormoterolUDP-glucuronosyltransferase 2B15enzyme
FormoterolSolute carrier family 22 member 1transporter
FormoterolSolute carrier family 22 member 4transporter
FormoterolOrganic cation/carnitine transporter 2transporter
HexoprenalineCalcium-activated potassium channel subunit alpha-1target
HexoprenalineBeta-2 adrenergic receptortarget
HigenamineBeta-2 adrenergic receptortarget
HigenamineBeta-1 adrenergic receptortarget
HigenamineLysine-specific histone demethylase 1Atarget
IndacaterolBeta-2 adrenergic receptortarget
IndacaterolCytochrome P450 3A4enzyme
IndacaterolUDP-glucuronosyltransferase 1A1enzyme
IndacaterolATP-dependent translocase ABCB1transporter
IsoetharineBeta-2 adrenergic receptortarget
IsoetharineBeta-1 adrenergic receptortarget
IsoprenalineBeta-1 adrenergic receptortarget
IsoprenalineBeta adrenergic receptortarget
IsoprenalineInterleukin-12 subunit betatarget
IsoprenalineCholinesteraseenzyme
IsoprenalineCatechol O-methyltransferaseenzyme
IsoprenalineAlbumincarrier
IsoprenalineCytochrome P450 1B1enzyme
IsoprenalineSuperoxide dismutase [Cu-Zn]target
IsoprenalineCytochrome P450 1A1enzyme
IsoprenalineBeta-3 adrenergic receptortarget
IsoprenalineBeta-2 adrenergic receptortarget
IsoxsuprineAlpha-1 adrenergic receptorstarget
IsoxsuprineBeta-2 adrenergic receptortarget
LevosalbutamolBeta-2 adrenergic receptortarget
LevosalbutamolSolute carrier organic anion transporter family member 1B1transporter
LevosalbutamolSolute carrier organic anion transporter family member 1B3transporter
LidamidineAlpha-2 adrenergic receptorstarget
MethoxyphenamineBeta-2 adrenergic receptortarget
MirabegronCytochrome P450 2D6enzyme
MirabegronUDP-glucuronosyltransferase 2B7enzyme
MirabegronUDP-glucuronosyltransferase 1A3enzyme
MirabegronUDP-glucuronosyltransferase 1A8enzyme
MirabegronSolute carrier family 22 member 1transporter
MirabegronBeta-3 adrenergic receptortarget
MirabegronCholinesteraseenzyme
MirabegronAlpha-1-acid glycoprotein 1carrier
MirabegronSolute carrier family 22 member 2transporter
MirabegronSolute carrier family 22 member 3transporter
MirabegronBeta-1 adrenergic receptortarget
MirabegronAlbumincarrier
MirabegronSolute carrier organic anion transporter family member 1A2transporter
MirabegronATP-dependent translocase ABCB1transporter
MirabegronCytochrome P450 3A4enzyme
NebivololBeta-1 adrenergic receptortarget
NebivololBeta-2 adrenergic receptortarget
NebivololCytochrome P450 3A4enzyme
NebivololAlbumincarrier
NebivololBeta-3 adrenergic receptortarget
NebivololCytochrome P450 2C19enzyme
NebivololCytochrome P450 2D6enzyme
NorepinephrineSynaptic vesicular amine transportertarget
NorepinephrineAlpha-1B adrenergic receptortarget
NorepinephrineSodium-dependent noradrenaline transportertransporter
NorepinephrinePOU domain, class 5, transcription factor 1transporter
NorepinephrineSolute carrier family 22 member 1transporter
NorepinephrineOrganic cation/carnitine transporter 2transporter
NorepinephrineSolute carrier family 22 member 3transporter
NorepinephrineSolute carrier family 22 member 2transporter
NorepinephrineBeta-3 adrenergic receptortarget
NorepinephrineBeta-2 adrenergic receptortarget
NorepinephrineAlpha-2B adrenergic receptortarget
NorepinephrineAlpha-2A adrenergic receptortarget
NorepinephrineAlpha-1D adrenergic receptortarget
NorepinephrineBeta-1 adrenergic receptortarget
NorepinephrineAlpha-1A adrenergic receptortarget
NorepinephrinePhenylalanine-4-hydroxylasetarget
NorepinephrineChromaffin granule amine transportertarget
NorepinephrineAlpha-2C adrenergic receptortarget
NylidrinCatechol O-methyltransferaseenzyme
NylidrinVoltage-dependent T-type calcium channel subunit alpha-1Itarget
NylidrinInterferon alpha/beta receptor 2target
NylidrinCytochrome P450 3A4enzyme
OlodaterolBeta-2 adrenergic receptortarget
OlodaterolCytochrome P450 2C9enzyme
OlodaterolCytochrome P450 2C8enzyme
OrciprenalineBeta-2 adrenergic receptortarget
OxyfedrineAldehyde dehydrogenase family 3 member A2target
OxyfedrineAldehyde dehydrogenase 1A1target
OxyfedrineBeta adrenergic receptortarget
PF-00610355Beta-2 adrenergic receptortarget
PhenylpropanolamineAmine oxidase [flavin-containing] Aenzyme
PhenylpropanolamineBeta-1 adrenergic receptortarget
PhenylpropanolamineBeta-2 adrenergic receptortarget
PhenylpropanolamineAlpha-2 adrenergic receptorstarget
PhenylpropanolamineSodium-dependent noradrenaline transportertarget
PhenylpropanolamineAlpha-1A adrenergic receptortarget
PhenylpropanolamineD(1A) dopamine receptortarget
PhenylpropanolamineTelomerase reverse transcriptasetarget
PirbuterolBeta-1 adrenergic receptortarget
PirbuterolBeta-2 adrenergic receptortarget
PrenalterolBeta-3 adrenergic receptortarget
ProcaterolBeta-2 adrenergic receptortarget
ProtokylolBeta-2 adrenergic receptortarget
ProtokylolBeta-1 adrenergic receptortarget
PseudoephedrineBeta-2 adrenergic receptortarget
PseudoephedrineAmine oxidase [flavin-containing] Aenzyme
PseudoephedrineBeta-1 adrenergic receptortarget
PseudoephedrineSodium-dependent dopamine transportertarget
PseudoephedrineSodium-dependent noradrenaline transportertarget
PseudoephedrineSodium-dependent serotonin transportertarget
PseudoephedrineNuclear factor of activated T-cells, cytoplasmic 1target
PseudoephedrineAlpha-1A adrenergic receptortarget
PseudoephedrineNuclear factor NF-kappa-B p105 subunittarget
Pseudoephedrineactivator protein 1target
PseudoephedrineInterleukin-2target
PseudoephedrineAlbumincarrier
PseudoephedrineSodium-dependent noradrenaline transportertransporter
PseudoephedrineSodium-dependent dopamine transportertransporter
PseudoephedrineSodium-dependent serotonin transportertransporter
PseudoephedrineD(2) dopamine receptortarget
PseudoephedrineAlpha-2A adrenergic receptortarget
PseudoephedrineTumor necrosis factortarget
RacepinephrineAlpha-2C adrenergic receptortarget
RacepinephrineBeta-3 adrenergic receptortarget
RacepinephrineAlpha-1D adrenergic receptortarget
RacepinephrineBeta-2 adrenergic receptortarget
RacepinephrineBeta-1 adrenergic receptortarget
RacepinephrineAlpha-2B adrenergic receptortarget
RacepinephrineAlpha-2A adrenergic receptortarget
RacepinephrineAlpha-1B adrenergic receptortarget
RacepinephrineAlpha-1A adrenergic receptortarget
RactopamineEstrogen receptortarget
ReproterolBeta-2 adrenergic receptortarget
RimiterolBeta-2 adrenergic receptortarget
RimiterolBeta-3 adrenergic receptortarget
RitobegronBeta-3 adrenergic receptortarget
RitodrineATP-sensitive potassium channeltarget
RitodrineMyosin light chain kinase, smooth muscletarget
RitodrineCalcium transporting ATPasestarget
RitodrineBeta-2 adrenergic receptortarget
Ritodrine6-phosphogluconate dehydrogenase, decarboxylatingenzyme
RitodrineSulfotransferase 1A1enzyme
RitodrineSulfotransferase 1A3enzyme
RitodrineBeta adrenergic receptortarget
RitodrineCalcium-activated potassium channeltarget
RitodrineSulfotransferase 1C4enzyme
RitodrineSulfotransferaseenzyme
RitodrineSulfotransferase 1C4target
SalmeterolBeta-2 adrenergic receptortarget
SalmeterolCytochrome P450 3A4enzyme
SalmeterolCytochrome P450 2C8enzyme
SalmeterolCytochrome P450 3A5enzyme
SalmeterolCytochrome P450 3A7enzyme
SalmeterolBeta-1 adrenergic receptortarget
SalmeterolSolute carrier family 22 member 3transporter
SalmeterolSolute carrier family 22 member 2transporter
SalmeterolBeta-3 adrenergic receptortarget
SalmeterolAlbumincarrier
Salmeterolalpha1-acid glycoproteincarrier
SalmeterolSolute carrier family 22 member 1transporter
SolabegronBeta-3 adrenergic receptortarget
TerbutalineBeta-1 adrenergic receptortarget
TerbutalineSolute carrier family 22 member 2transporter
TerbutalineOrganic cation/carnitine transporter 2transporter
TerbutalineUDP-glucuronosyltransferases (UGTs)enzyme
TerbutalineSulfotransferaseenzyme
TerbutalineBeta-2 adrenergic receptortarget
TerbutalineCholinesteraseenzyme
TerbutalineBeta-3 adrenergic receptortarget
TretoquinolBeta-2 adrenergic receptortarget
TulobuterolBeta-2 adrenergic receptortarget
VibegronBeta-3 adrenergic receptortarget
VibegronCytochrome P450 3A4enzyme
VibegronATP-dependent translocase ABCB1transporter
VilanterolCytochrome P450 3A4enzyme
VilanterolBeta-2 adrenergic receptortarget
VilanterolATP-dependent translocase ABCB1transporter
XamoterolBeta-1 adrenergic receptortarget
XamoterolBeta-3 adrenergic receptortarget