Central alpha-2 Adrenergic Agonist

Name
Central alpha-2 Adrenergic Agonist
Accession Number
DBCAT003378
Description

Not Available

Drugs
DrugDrug Description
ClonidineAn alpha-2 adrenergic agonist used to treat hypertension and severe cancer pain, among other conditions, and to treat withdrawal symptoms from various substances. It is also used to aid in the diagnosis of pheochromocytoma and to prevent migraines.
DexmedetomidineAn alpha-2 agonist used for sedation during various procedures.
GuanabenzAn alpha-2 adrenergic agonist used to treat hypertension.
GuanfacineAn alpha-2A adrenergic receptor agonist used to treat ADHD.
LofexidineA centrally acting alpha2-adrenergic agonist used for the symptomatic treatment of acute opioid withdrawal syndrome to facilitate abrupt opioid discontinuation in adults.
MethyldopaA centrally-acting alpha-2 adrenergic agonist used to manage hypertension alone or in combination with hydrochlorothiazide, and to treat hypertensive crises.
TizanidineAn alpha-2 adrenergic agonist used for the short-term treatment of muscle spasticity.
Drugs & Drug Targets
DrugTargetType
ClonidineAlpha-2A adrenergic receptortarget
ClonidineCytochrome P450 2D6enzyme
ClonidineAlpha-2B adrenergic receptortarget
ClonidineAlpha-2C adrenergic receptortarget
ClonidineSolute carrier family 22 member 3transporter
ClonidineOrganic cation/carnitine transporter 2transporter
ClonidineSolute carrier family 22 member 4transporter
ClonidineCytochrome P450 1A2enzyme
ClonidineCytochrome P450 3A4enzyme
ClonidineCytochrome P450 1A1enzyme
ClonidineCytochrome P450 3A5enzyme
ClonidineAlpha-1A adrenergic receptortarget
ClonidineAlpha-1B adrenergic receptortarget
ClonidineAlpha-1D adrenergic receptortarget
ClonidineAlbumincarrier
ClonidineAmine oxidase [copper-containing] 3target
ClonidineAlpha-2 adrenergic receptorstarget
DexmedetomidineAlpha-2 adrenergic receptorstarget
DexmedetomidineCytochrome P450 2D6enzyme
DexmedetomidineCytochrome P450 1A1enzyme
DexmedetomidineCytochrome P450 1A2enzyme
DexmedetomidineAlpha-2A adrenergic receptortarget
DexmedetomidineCytochrome P450 2E1enzyme
GuanabenzAlpha-2 adrenergic receptorstarget
GuanabenzAlpha-2B adrenergic receptortarget
GuanabenzCytochrome P450 1A2enzyme
GuanabenzAlpha-2A adrenergic receptortarget
GuanfacineAlpha-2 adrenergic receptorstarget
GuanfacineSolute carrier family 22 member 2transporter
GuanfacineSolute carrier family 22 member 1transporter
GuanfacineMultidrug and toxin extrusion protein 1transporter
GuanfacineAlpha-2B adrenergic receptortarget
GuanfacineCytochrome P450 3A4enzyme
GuanfacineCytochrome P450 2C19enzyme
GuanfacineAlpha-2A adrenergic receptortarget
LofexidineAlpha-2 adrenergic receptorstarget
LofexidineAlpha-2A adrenergic receptortarget
LofexidineAlpha-1A adrenergic receptortarget
Lofexidine5-hydroxytryptamine receptor 1Atarget
Lofexidine5-hydroxytryptamine receptor 7target
Lofexidine5-hydroxytryptamine receptor 2Ctarget
Lofexidine5-hydroxytryptamine receptor 1Dtarget
LofexidineCytochrome P450 2D6enzyme
LofexidineCytochrome P450 1A2enzyme
LofexidineCytochrome P450 2C19enzyme
LofexidineATP-binding cassette sub-family B member 5transporter
LofexidineMultidrug and toxin extrusion protein 1transporter
MethyldopaSulfotransferaseenzyme
MethyldopaDopamine beta-hydroxylaseenzyme
MethyldopaPhenylethanolamine N-methyltransferaseenzyme
MethyldopaAromatic-L-amino-acid decarboxylaseenzyme
MethyldopaD(2) dopamine receptortarget
MethyldopaAlpha-2 adrenergic receptorstarget
MethyldopaAromatic-L-amino-acid decarboxylasetarget
MethyldopaSolute carrier family 15 member 1transporter
MethyldopaCatechol O-methyltransferaseenzyme
MethyldopaAlbumincarrier
MethyldopaAlpha-2A adrenergic receptortarget
TizanidineAlpha-1 adrenergic receptorstarget
TizanidineNischarintarget
TizanidineCytochrome P450 1A2enzyme
TizanidineAlpha-2 adrenergic receptorstarget