Estrogen Agonist/Antagonist

All categories

Name: Estrogen Agonist/Antagonist
Accession Number: DBCAT003358
Description: Not Available
Drugs: Drug Drug Description
Bazedoxifene A selective estrogen receptor modulator (SERM) used to treat moderate to severe vasomotor symptoms in menopause and osteoporosis alone or in combination with conjugated estrogens.
Clomifene A medication used to induce ovulation.
Ospemifene A non-hormonal estrogen receptor modulator (SERM) used to treat moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause.
Raloxifene A selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women.
Tamoxifen A selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
Toremifene A first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.
Drugs & Drug Targets: Drug Target Type
Bazedoxifene Estrogen receptor target
Bazedoxifene UDP-glucuronosyltransferase 1A10 enzyme
Bazedoxifene UDP-glucuronosyltransferase 1A8 enzyme
Bazedoxifene Estrogen receptor beta target
Bazedoxifene UDP-glucuronosyltransferase 1A4 enzyme
Bazedoxifene Estrogen receptor target
Clomifene Estrogen receptor beta target
Clomifene Steroid 17-alpha-hydroxylase/17,20 lyase enzyme
Clomifene ATP-dependent translocase ABCB1 transporter
Clomifene Estrogen receptor target
Ospemifene Estrogen receptor target
Ospemifene Cytochrome P450 2D6 enzyme
Ospemifene Cytochrome P450 2B6 enzyme
Ospemifene Cytochrome P450 2C19 enzyme
Ospemifene Cytochrome P450 2C9 enzyme
Ospemifene Cytochrome P450 3A4 enzyme
Ospemifene Estrogen receptor target
Raloxifene ATP-binding cassette sub-family C member 3 transporter
Raloxifene ATP-binding cassette sub-family C member 4 transporter
Raloxifene UDP-glucuronosyltransferase 1A10 enzyme
Raloxifene UDP-glucuronosyltransferase 1A8 enzyme
Raloxifene Estrogen receptor beta target
Raloxifene Aldehyde oxidase enzyme
Raloxifene Cytochrome P450 2C8 enzyme
Raloxifene Cytochrome P450 2B6 enzyme
Raloxifene Aromatase enzyme
Raloxifene Cytochrome P450 3A4 enzyme
Raloxifene Serpin B9 target
Raloxifene Trefoil factor 1 target
Raloxifene UDP-glucuronosyltransferase 1A1 enzyme
Raloxifene Albumin carrier
Raloxifene Alpha-1-acid glycoprotein 1 carrier
Raloxifene Solute carrier organic anion transporter family member 1B1 transporter
Raloxifene Solute carrier organic anion transporter family member 1B3 transporter
Raloxifene ATP-dependent translocase ABCB1 transporter
Raloxifene Broad substrate specificity ATP-binding cassette transporter ABCG2 transporter
Raloxifene ATP-binding cassette sub-family C member 2 transporter
Raloxifene Estrogen receptor target
Tamoxifen Cytochrome P450 2C19 enzyme
Tamoxifen Flavin-containing monooxygenase 1 enzyme
Tamoxifen Flavin-containing monooxygenase 3 enzyme
Tamoxifen Cytochrome P450 3A7 enzyme
Tamoxifen Cytochrome P450 1B1 enzyme
Tamoxifen Broad substrate specificity ATP-binding cassette transporter ABCG2 transporter
Tamoxifen Aromatase enzyme
Tamoxifen Cytochrome P450 2A6 enzyme
Tamoxifen Cytochrome P450 2E1 enzyme
Tamoxifen UDP-glucuronosyltransferase 1A10 enzyme
Tamoxifen Sulfotransferase 1A1 enzyme
Tamoxifen ATP-binding cassette sub-family C member 2 transporter
Tamoxifen 3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase target
Tamoxifen Protein kinase C target
Tamoxifen Androgen receptor target
Tamoxifen Voltage-gated inwardly rectifying potassium channel KCNH2 target
Tamoxifen Nuclear receptor subfamily 1 group I member 2 target
Tamoxifen Estrogen-related receptor gamma target
Tamoxifen Sex hormone-binding globulin target
Tamoxifen Bile salt export pump transporter
Tamoxifen Thyroxine-binding globulin carrier
Tamoxifen Sulfotransferase 2A1 enzyme
Tamoxifen Cytochrome P450 1A2 enzyme
Tamoxifen UDP-glucuronosyltransferase 2B7 enzyme
Tamoxifen UDP-glucuronosyltransferase 2B17 enzyme
Tamoxifen Sulfotransferase 1E1 enzyme
Tamoxifen Phospholipid-transporting ATPase ABCA1 transporter
Tamoxifen Mitogen-activated protein kinase 8 target
Tamoxifen Albumin carrier
Tamoxifen Cytochrome P450 1A1 enzyme
Tamoxifen Cytochrome P450 3A5 enzyme
Tamoxifen Liver carboxylesterase 1 enzyme
Tamoxifen Cytochrome P450 2B6 enzyme
Tamoxifen Cytochrome P450 2C8 enzyme
Tamoxifen Cytochrome P450 2D6 enzyme
Tamoxifen Cytochrome P450 3A4 enzyme
Tamoxifen Cytochrome P450 2C9 enzyme
Tamoxifen Estrogen receptor beta target
Tamoxifen Estrogen receptor target
Tamoxifen ATP-dependent translocase ABCB1 transporter
Toremifene Sex hormone-binding globulin target
Toremifene Cytochrome P450 1A1 enzyme
Toremifene ATP-dependent translocase ABCB1 transporter
Toremifene Cytochrome P450 3A4 enzyme
Toremifene Estrogen receptor target
Toremifene Estrogen receptor target

Drug	Drug Description
Bazedoxifene	A selective estrogen receptor modulator (SERM) used to treat moderate to severe vasomotor symptoms in menopause and osteoporosis alone or in combination with conjugated estrogens.
Clomifene	A medication used to induce ovulation.
Ospemifene	A non-hormonal estrogen receptor modulator (SERM) used to treat moderate to severe dyspareunia, a symptom of vulvar and vaginal atrophy, due to menopause.
Raloxifene	A selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women.
Tamoxifen	A selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
Toremifene	A first generation nonsteroidal selective estrogen receptor modulator used to treat certain breast cancers.

Estrogen Agonist/Antagonist

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