Roblitinib

DB16845InvestigationalSmall molecule

Roblitinib: Overview.

Mechanism: Pharmacologically active on Fibroblast growth factor receptor 4
Curator reviewed
Formula / weight: C₂₅H₃₀N₈O₄ · 506.567 g/mol (avg)
Code names: FGF-401

Resolves to

Compound

Structure

InChIKeyBHKDKKZMPODMIQ-UHFFFAOYSA-NSMILESCOCCNC1=CC(NC(=O)N2CCCC3=CC(CN4CCN(C)CC4=O)=C(C=O)N=C23)=NC=C1C#N

Targets

What you can answer from here — as of June 15, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1Clinical trialPhase, status and sponsor resolved per trial

4+ReferencesStructured and connected to the statements they support

Which drugs share a target with Roblitinib, and which of those have an active Phase 3 trial?

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