RS-39604

DB17050ExperimentalSmall molecule

RS-39604 is a selective 5-HT4 receptor antagonist.

Mechanism: Pharmacologically active on 5-hydroxytryptamine receptor 4
Curator reviewed
Formula / weight: C₂₆H₃₆ClN₃O₆S · 554.1 g/mol (avg)
Also known as: Methanesulfonamide, n-(2-(4-(3-(4-amino-5-chloro-2-((3,5-dimethoxyphenyl)methoxy)phenyl)-3-oxopropyl)-1-piperidinyl)ethyl)-
Code names: RS-39604

Resolves to

Compound

Structure

InChIKeyBKVIWGRFRKLFIO-UHFFFAOYSA-NSMILESCOC1=CC(OC)=CC(COC2=CC(N)=C(Cl)C=C2C(=O)CCC2CCN(CCNS(C)(=O)=O)CC2)=C1

Targets

What you can answer from here — as of July 17, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

6+ReferencesStructured and connected to the statements they support

Which drugs share a target with RS-39604, and which of those have an active Phase 3 trial?

Create a free account or log in to explore the full data card.