| DB00604 | Cisapride | approved, investigational, withdrawn | yes | agonist | Details |
| DB01079 | Tegaserod | approved, investigational, withdrawn | yes | antagonistpartial agonist | Details |
| DB04873 | Piboserod | investigational | unknown | | Details |
| DB04917 | Renzapride | investigational | unknown | | Details |
| DB12702 | Velusetrag | investigational | unknown | | Details |
| DB05905 | TD-2749 | investigational | unknown | | Details |
| DB06422 | Ticalopride | investigational | unknown | | Details |
| DB06480 | Prucalopride | approved | yes | agonist | Details |
| DB05542 | Naronapride | investigational | unknown | agonist | Details |
| DB01233 | Metoclopramide | approved, investigational | yes | agonist | Details |
| DB00904 | Ondansetron | approved, withdrawn | unknown | agonist | Details |
| DB08810 | Cinitapride | investigational | unknown | agonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | agonist | Details |