Unesbulin

DB18080InvestigationalSmall molecule

Unesbulin: Overview.

Chemical structure of Unesbulin
Formula / weight
C19H13F5N6 · 420.347 g/mol (avg)
Also known as
4,6-pyrimidinediamine, 5-fluoro-2-(6-fluoro-2-methyl-1h-benzimidazol-1-yl)-n4-(4-(trifluoromethyl)phenyl)- · 5-fluoro-2-(6-fluoro-2-methyl-1h-benzimidazol-1-yl)-n4-(4-(trifluoromethyl)phenyl)-4,6-pyrimidinediamine · 5-fluoro-2-(6-fluoro-2-methyl-1h-benzo(d)imidazole-1-yl)-n4-(4-(trifluoromethyl)phenyl)pyrimidine-4,6-diamine · 5-fluoro-2-(6-fluoro-2-methyl-1H-benzo[d]imidazole-1-yl)-N4-(4-(trifluoromethyl)phenyl)pyrimidine-4,6-diamine · Bmi1 inhibitor ptc596
Code names
PTC-596

Resolves to

Compound
UNIIZ4HZ70S62QCAS1610964-64-1ChEMBLCHEMBL4594353
Structure
InChIKeyTWLWOOPCEXYVBE-UHFFFAOYSA-NSMILESCC1=NC2=CC=C(F)C=C2N1C1=NC(N)=C(F)C(NC2=CC=C(C=C2)C(F)(F)F)=N1
Targets
P35226BMI1

What you can answer from here — as of April 23, 2025

1Protein targetEach mapped to UniProt, with action and pharmacological action
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5Clinical trialsPhase, status and sponsor resolved per trial
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1+ReferenceStructured and connected to the statements they support
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Which drugs share a target with Unesbulin, and which of those have an active Phase 3 trial?

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