Velzatinib

DB18087InvestigationalSmall molecule

Velzatinib: Overview.

Mechanism: Pharmacologically active on Mast/stem cell growth factor receptor Kit
Curator reviewed
Formula / weight: C₂₉H₃₂N₈O · 508.63 g/mol (avg)
Code names: IDRX-42

Resolves to

Compound

Structure

InChIKeyLVMAULGVWBINFP-UHFFFAOYSA-NSMILESCN1C=C(C=N1)C1=CC=C(CNC2=CC(=NC=N2)C2=CN=C3C=C(OCCCN4CCCC4)C=CN23)C=C1

Targets

What you can answer from here — as of September 25, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

6Clinical trialsPhase, status and sponsor resolved per trial

2+ReferencesStructured and connected to the statements they support

Which drugs share a target with Velzatinib, and which of those have an active Phase 3 trial?

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