| DB00398 | Sorafenib | approved, investigational | yes | antagonist | Details |
| DB00619 | Imatinib | approved | yes | antagonist | Details |
| DB01254 | Dasatinib | approved, investigational | yes | antagonist | Details |
| DB01268 | Sunitinib | approved, investigational | yes | inhibitor | Details |
| DB01962 | Phosphonotyrosine | experimental | unknown | | Details |
| DB04868 | Nilotinib | approved, investigational | unknown | antagonist | Details |
| DB12742 | Amuvatinib | investigational | unknown | | Details |
| DB05146 | XL820 | investigational | unknown | | Details |
| DB06080 | Linifanib | investigational | unknown | | Details |
| DB05913 | OSI-930 | investigational | unknown | | Details |
| DB06589 | Pazopanib | approved | yes | inhibitor | Details |
| DB06595 | Midostaurin | approved, investigational | unknown | antagonistinhibitor | Details |
| DB08896 | Regorafenib | approved | yes | inhibitor | Details |
| DB08901 | Ponatinib | approved, investigational | unknown | inhibitor | Details |
| DB09078 | Lenvatinib | approved, investigational | yes | inhibitor | Details |
| DB09103 | Ancestim | approved, investigational, withdrawn | yes | agonist | Details |
| DB12010 | Fostamatinib | approved, investigational | unknown | inhibitor | Details |
| DB12147 | Erdafitinib | approved, investigational | unknown | substrate | Details |
| DB12978 | Pexidartinib | approved, investigational | unknown | inhibitor | Details |
| DB15233 | Avapritinib | approved, investigational | unknown | inhibitor | Details |
| DB14840 | Ripretinib | approved | yes | inhibitor | Details |
| DB11800 | Tivozanib | approved, investigational | yes | inhibitor | Details |