Opelconazole

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DB18251InvestigationalSmall molecule

Opelconazole: Overview.

Mechanism: Pharmacologically active on Lanosterol 14-alpha demethylase
Curator reviewed
Formula / weight: C₃₈H₃₇F₃N₆O₃ · 682.748 g/mol (avg)
Also known as: D-threo-pentitol, 2,5-anhydro-1,3,4-trideoxy-2-c-(2,4-difluorophenyl)-4-((4-(4-(4-(((4-fluorophenyl)amino)carbonyl)phenyl)-1-piperazinyl)-2-methylphenoxy)methyl)-1-(1h-1,2,4-triazol-1-yl)- · Opelconazole(inn)
Code names: PC-945

Resolves to

Compound

UNII45LU8Q6ASUCAS1931946-73-4ChEMBLCHEMBL4650362

Structure

InChIKeyOSAMZQJKSCAOHA-CWRQMEKBSA-NSMILESCC1=CC(=CC=C1OC[C@@H]1CO[C@](CN2C=NC=N2)(C1)C1=CC=C(F)C=C1F)N1CCN(CC1)C1=CC=C(C=C1)C(=O)NC1=CC=C(F)C=C1

Targets

P10613ERG11

What you can answer from here — as of July 09, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

6Clinical trialsPhase, status and sponsor resolved per trial

4+ReferencesStructured and connected to the statements they support

Which drugs share a target with Opelconazole, and which of those have an active Phase 3 trial?

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