Flurpiridaz F-18

Identification

Generic Name
Flurpiridaz F-18
DrugBank Accession Number
DB18773
Background

Not Available

Type
Small Molecule
Groups
Investigational
Structure
Weight
Average: 367.84
Monoisotopic: 367.1328329
Chemical Formula
C18H22ClFN2O3
Synonyms
  • 2-tert-butyl-4-chloro-5-((4-((2-(18f)fluoroethoxy)methyl)phenyl)methoxy)pyridazin-3(2h)-one
  • 3(2h)-pyridazinone, 4-chloro-2-(1,1-dimethylethyl)-5-((4-((2-(fluoro-(sup 18)f)ethoxy)methyl)phenyl)methoxy)-
  • 3(2h)-pyridazinone, 4-chloro-2-(1,1-dimethylethyl)-5-((4-((2-(fluoro-18f)ethoxy)methyl)phenyl)methoxy)-
  • 4-chloro-2-(1,1-dimethylethyl)-5-((4-((2-((sup 18)f)fluoroethoxy)methyl)phenyl) methoxy)pyridazin-3(2h)-one
  • Flurpiridaz (18f)
  • Flurpiridaz f 18
  • Flurpiridaz, F-18
External IDs
  • BMS 747158-02
  • BMS-747158
  • BMS-747158-02

Pharmacology

Indication

Not Available

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Pharmacodynamics

Not Available

Mechanism of action
Not Available
Absorption

Not Available

Volume of distribution

Not Available

Protein binding

Not Available

Metabolism
Not Available
Route of elimination

Not Available

Half-life

Not Available

Clearance

Not Available

Adverse Effects
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Toxicity

Not Available

Pathways
Not Available
Pharmacogenomic Effects/ADRs
Not Available

Interactions

Drug Interactions
This information should not be interpreted without the help of a healthcare provider. If you believe you are experiencing an interaction, contact a healthcare provider immediately. The absence of an interaction does not necessarily mean no interactions exist.
Not Available
Food Interactions
Not Available

Categories

Drug Categories
Classification
Not classified
Affected organisms
Not Available

Chemical Identifiers

UNII
TY3V24C029
CAS number
863887-89-2
InChI Key
RMXZKEPDYBTFOS-LRFGSCOBSA-N
InChI
InChI=1S/C18H22ClFN2O3/c1-18(2,3)22-17(23)16(19)15(10-21-22)25-12-14-6-4-13(5-7-14)11-24-9-8-20/h4-7,10H,8-9,11-12H2,1-3H3/i20-1
IUPAC Name
SMILES
CC(C)(C)N1N=CC(OCC2=CC=C(COCC[18F])C=C2)=C(Cl)C1=O

References

General References
Not Available
ChemSpider
9580860
ChEMBL
CHEMBL2107799
ZINC
ZINC000100529282

Clinical Trials

Clinical Trials
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PhaseStatusPurposeConditionsCountStart DateWhy Stopped100+ additional columns
3CompletedDiagnosticCoronary Artery Disease (CAD)1somestatusstop reasonjust information to hide
3WithdrawnDiagnosticCoronary Artery Disease (CAD)1somestatusstop reasonjust information to hide
2CompletedDiagnosticCoronary Artery Disease (CAD) / Ischemic Heart Disease1somestatusstop reasonjust information to hide
2CompletedDiagnosticIschemia1somestatusstop reasonjust information to hide
1CompletedDiagnosticCoronary Artery Disease (CAD)1somestatusstop reasonjust information to hide

Pharmacoeconomics

Manufacturers
Not Available
Packagers
Not Available
Dosage Forms
Not Available
Prices
Not Available
Patents
Not Available

Properties

State
Not Available
Experimental Properties
Not Available
Predicted Properties
PropertyValueSource
Predicted ADMET Features
Not Available

Spectra

Mass Spec (NIST)
Not Available
Spectra
Not Available
Chromatographic Properties
Collision Cross Sections (CCS)
Not Available

Drug created at June 19, 2024 19:42 / Updated at June 21, 2024 20:33