Opevesostat

DB18818InvestigationalSmall molecule

Opevesostat: Overview.

Mechanism: Pharmacologically active on Cholesterol side-chain cleavage enzyme, mitochondrial
Curator reviewed
Formula / weight: C₂₁H₂₆N₂O₅S · 418.51 g/mol (avg)
Code names: MK-5684 · ODM-208

Resolves to

Compound

Structure

InChIKeyLHVKCOBGLZGRQZ-UHFFFAOYSA-NSMILESCS(=O)(=O)N1CCC(COC2=COC(CN3CC4=CC=CC=C4C3)=CC2=O)CC1

Targets

What you can answer from here — as of July 09, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

12Clinical trialsPhase, status and sponsor resolved per trial

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with Opevesostat, and which of those have an active Phase 3 trial?

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