Telenzepine

DB19508InvestigationalSmall molecule

Telenzepine is a small molecule drug. The usage of the INN stem '-zepine' in the name indicates that Telenzepine is a tricyclic compound. Telenzepine is under investigation in clinical trial... Telenzepine is under investigation in clinical trial NCT01155531 (Safety & Tolerability of a Combination of Antidepressant and Peptic Ulcer Drug in Overweight Healthy Subjects).

Chemical structure of Telenzepine
Formula / weight
C19H22N4O2S · 370.47 g/mol (avg)
Code names
NSC-758679

Resolves to

Compound
UNII0990EG3K10CAS80880-90-6ChEMBLCHEMBL253978ChEBI92110PubChem5387
Structure
InChIKeyVSWPGAIWKHPTKX-UHFFFAOYSA-NSMILESCN1CCN(CC(=O)N2C3=C(C)SC=C3C(=O)NC3=CC=CC=C23)CC1
Targets
P11229CHRM1

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
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1Clinical trialPhase, status and sponsor resolved per trial
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1+ReferenceStructured and connected to the statements they support
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Which drugs share a target with Telenzepine, and which of those have an active Phase 3 trial?

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