Temelastine

DB20506ExperimentalSmall molecule

Temelastine is a small molecule drug. The usage of the INN stem '-astine' in the name indicates that Temelastine is a antihistaminic. Temelastine has a monoisotopic molecular weight of 441.12...

Mechanism: Pharmacologically active on Histamine H1 receptor
Curator reviewed
Formula / weight: C₂₁H₂₄BrN₅O · 442.361 g/mol (avg)
Code names: SK&F-93944

Resolves to

Compound

UNIIBF6IGI53XHCAS86181-42-2ChEMBLCHEMBL70598ChEBI180882

Structure

InChIKeyOGEAASSLWZDQBM-UHFFFAOYSA-NSMILESCC1=NC=C(CC2=CNC(NCCCCC3=NC=C(Br)C=C3C)=NC2=O)C=C1

Targets

P35367HRH1

What you can answer from here — as of September 16, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

2+ReferencesStructured and connected to the statements they support

Which drugs share a target with Temelastine, and which of those have an active Phase 3 trial?

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