Setoperone

DB20520ExperimentalSmall molecule

Setoperone is a small molecule drug. The usage of the INN stem '-perone' in the name indicates that Setoperone is a tranquillizer, neuroleptic, 4'-fluoro-4-piperidinobutyrophenone derivative. Setoperone has a monoisotopic molecular...

Mechanism: Pharmacologically active on Dopamine receptor D2 and 5-hydroxytryptamine receptor 2
Curator reviewed
Formula / weight: C₂₁H₂₄FN₃O₂S · 401.5 g/mol (avg)
Code names: R-52245

Resolves to

Compound

UNIIBQ67CS3Q3ECAS86487-64-1ChEMBLCHEMBL2105437ChEBI229894PubChem68604

Structure

InChIKeyRBGAHDDQSRBDOG-UHFFFAOYSA-NSMILESCC1=C(CCN2CCC(CC2)C(=O)C2=CC=C(F)C=C2)C(=O)N2CCSC2=N1

Targets

P14416DRD2

What you can answer from here — as of September 23, 2026

2Protein targetsEach mapped to UniProt, with action and pharmacological action

Listed above

3+ReferencesStructured and connected to the statements they support

Which drugs share a target with Setoperone, and which of those have an active Phase 3 trial?

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