Terlakiren

DB20615ExperimentalSmall molecule

Terlakiren is a small molecule drug. The usage of the INN stem '-kiren' in the name indicates that Terlakiren is a renin inhibitor. Terlakiren has a monoisotopic molecular weight of...

Chemical structure of Terlakiren
Formula / weight
C31H48N4O7S · 620.81 g/mol (avg)
Code names
CP-80,794

Resolves to

Structure
InChIKeyUZQBKCWYZBHBOW-YIPNQBBMSA-NSMILESCSC[C@H](NC(=O)[C@H](CC1=CC=CC=C1)NC(=O)N1CCOCC1)C(=O)N[C@@H](CC1CCCCC1)[C@@H](O)C(=O)OC(C)C
Targets

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
Listed above
3+ReferencesStructured and connected to the statements they support
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Which drugs share a target with Terlakiren, and which of those have an active Phase 3 trial?

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