Rafabegron

DB20910ExperimentalSmall molecule

Rafabegron is a small molecule drug. The usage of the INN stem '-begron' in the name indicates that Rafabegron is a β3 adrenoreceptor agonists. Rafabegron has a monoisotopic molecular weight...

Mechanism: Pharmacologically active on Beta-3 adrenergic receptor
Curator reviewed
Formula / weight: C₂₁H₂₃ClN₂O₄ · 402.88 g/mol (avg)
Code names: AD-9677 · TAK-677

Resolves to

Compound

UNIILN3E1Q0SU2CAS244081-42-3ChEMBLCHEMBL279260ChEBI748056PubChem5493324

Structure

InChIKeyFHEYFIGWYQJVDR-ACJLOTCBSA-NSMILESC[C@H](CC1=CNC2=C(OCC(O)=O)C=CC=C12)NC[C@H](O)C1=CC(Cl)=CC=C1

Targets

P13945ADRB3

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

5+ReferencesStructured and connected to the statements they support

Which drugs share a target with Rafabegron, and which of those have an active Phase 3 trial?

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