| DB00368 | Norepinephrine | approved | yes | agonist | Details |
| DB00571 | Propranolol | approved, investigational | unknown | antagonist | Details |
| DB05395 | Amibegron | investigational | unknown | | Details |
| DB06262 | Droxidopa | approved, investigational | yes | agonist | Details |
| DB06190 | Solabegron | investigational | unknown | agonist | Details |
| DB01288 | Fenoterol | approved, investigational | unknown | agonist | Details |
| DB01407 | Clenbuterol | approved, investigational, vet_approved | unknown | agonist | Details |
| DB01102 | Arbutamine | approved | unknown | agonist | Details |
| DB01064 | Isoprenaline | approved, investigational | yes | agonist | Details |
| DB08807 | Bopindolol | experimental | unknown | | Details |
| DB08808 | Bupranolol | experimental | unknown | antagonist | Details |
| DB01363 | Ephedra sinica root | nutraceutical | yes | agonist | Details |
| DB08893 | Mirabegron | approved | yes | agonist | Details |
| DB01001 | Salbutamol | approved, vet_approved | unknown | | Details |
| DB00866 | Alprenolol | experimental, withdrawn | unknown | antagonist | Details |
| DB00983 | Formoterol | approved, investigational | unknown | agonist | Details |
| DB00938 | Salmeterol | approved | unknown | inverse agonist | Details |
| DB00871 | Terbutaline | approved | unknown | agonist | Details |
| DB00960 | Pindolol | approved, investigational | unknown | agonist | Details |
| DB01580 | Oxprenolol | approved | unknown | | Details |
| DB11124 | Racepinephrine | approved | yes | agonist | Details |
| DB04846 | Celiprolol | approved, investigational | unknown | agonist | Details |
| DB04861 | Nebivolol | approved, investigational | unknown | agonist | Details |
| DB14895 | Vibegron | approved, investigational | yes | agonist | Details |
| DB00320 | Dihydroergotamine | approved, investigational | unknown | agonist | Details |