Befetupitant

DB21149ExperimentalSmall molecule

Befetupitant is a small molecule drug. The usage of the INN stem '-pitant' in the name indicates that Befetupitant is a neurokinin NK1​ (substance P) receptor antagonist. Befetupitant has a... Befetupitant has a monoisotopic molecular weight of 565.22 Da.

Chemical structure of Befetupitant
Formula / weight
C29H29F6N3O2 · 565.56 g/mol (avg)
Code names
RO 67-5930 · RO 67-5930/000

Resolves to

Compound
UNIIRSH7NDI7MICAS290296-68-3ChEMBLCHEMBL204694ChEBI748735PubChem6450815
Structure
InChIKeyZGNPLCMMVKCTHM-UHFFFAOYSA-NSMILESCN(C(=O)C(C)(C)C1=CC(=CC(=C1)C(F)(F)F)C(F)(F)F)C1=C(C=C(N=C1)N1CCOCC1)C1=C(C)C=CC=C1
Targets
P25103TACR1

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
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3+ReferencesStructured and connected to the statements they support
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