Lomeguatrib

DB21175ExperimentalSmall molecule

Lomeguatrib is a small molecule drug. Lomeguatrib has a monoisotopic molecular weight of 324.96 Da.

Mechanism: Pharmacologically active on Methylated-DNA--protein-cysteine methyltransferase
Curator reviewed
Formula / weight: C₁₀H₈BrN₅OS · 326.17 g/mol (avg)

Resolves to

Compound

Structure

InChIKeyJUJPKFNFCWJBCX-UHFFFAOYSA-NSMILESNC1=NC(OCC2=CC(Br)=CS2)=C2NC=NC2=N1

Targets

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

6+ReferencesStructured and connected to the statements they support

Which drugs share a target with Lomeguatrib, and which of those have an active Phase 3 trial?

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