Bamirastine

DB21186ExperimentalSmall molecule

Bamirastine is a small molecule drug. The usage of the INN stem '-astine' in the name indicates that Bamirastine is a antihistaminic. Bamirastine has a monoisotopic molecular weight of 527.29...

Mechanism: Pharmacologically active on Histamine H1 receptor
Curator reviewed
Formula / weight: C₃₁H₃₇N₅O₃ · 527.669 g/mol (avg)
Code names: TAK-427

Resolves to

Compound

UNIISIG10953FNCAS215529-47-8ChEMBLCHEMBL2107732ChEBI752829PubChem9806921

Structure

InChIKeyWTBRUSNNZKWTMI-UHFFFAOYSA-NSMILESCC(C)(C(O)=O)C1=CN2N=C(NCCCN3CCC(CC3)OC(C3=CC=CC=C3)C3=CC=CC=C3)C=CC2=N1

Targets

P35367HRH1

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with Bamirastine, and which of those have an active Phase 3 trial?

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