Setipafant

DB21252ExperimentalSmall molecule

Setipafant is a small molecule drug. The usage of the INN stem '-pafant' in the name indicates that Setipafant is a platelet-activating factor antagonist. Setipafant has a monoisotopic molecular weight...

Formula / weight: C₂₆H₂₃ClN₆O₂S · 519.02 g/mol (avg)

Resolves to

Compound

UNIIUFN2Q54HS6CAS132418-35-0ChEMBLCHEMBL2107078ChEBI752419PubChem65968

Structure

InChIKeyDDJKTQDAEYPACV-UHFFFAOYSA-NSMILESCOC1=CC=C(NC(=O)N2CCC3=C(C2)SC2=C3C(=NCC3=NN=C(C)N23)C2=CC=CC=C2Cl)C=C1

Targets

P25105PTAFR

What you can answer from here — as of September 23, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with Setipafant, and which of those have an active Phase 3 trial?

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