Lupitidine

DB21334ExperimentalSmall molecule

Lupitidine is a small molecule drug. The usage of the INN stem '-tidine' in the name indicates that Lupitidine is a histamine- H2-receptor antagonist, cimetidine derivative. Lupitidine has a monoisotopic...

Mechanism: Pharmacologically active on Histamine H2 receptor
Curator reviewed
Formula / weight: C₂₁H₂₇N₅O₂S · 413.54 g/mol (avg)
Code names: CM-10

Resolves to

Compound

UNIIWF028DWK9NCAS83903-06-4ChEMBLCHEMBL69178

Structure

InChIKeyIKEHSFKMCULMKJ-UHFFFAOYSA-NSMILESCN(C)CC1=CC=C(CSCCNC2=NC=C(CC3=CC=C(C)N=C3)C(=O)N2)O1

Targets

P25021HRH2

What you can answer from here — as of September 13, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1+ReferenceStructured and connected to the statements they support

Which drugs share a target with Lupitidine, and which of those have an active Phase 3 trial?

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