Amcenestrant

DB21753InvestigationalSmall molecule

Amcenestrant: Overview.

Mechanism
Curator reviewed
Also known as
5H-BENZOCYCLOHEPTENE-3-CARBOXYLIC ACID, 8-(2,4-DICHLOROPHENYL)-9-(4-(((3S)-1-(3-FLUOROPROPYL)-3-PYRROLIDINYL)OXY)PHENYL)-6,7-DIHYDRO- · 8-(2,4-DICHLOROPHENYL)-9-(4-(((3S)-1-(3-FLUOROPROPYL)-3-PYRROLIDINYL)OXY)PHENYL)-6,7-DIHYDRO-5H-BENZOCYCLOHEPTENE-3-CARBOXYLIC ACID · 8-(2,4-DICHLOROPHENYL)-9-(4-(((3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL)OXY)PHENYL)-6,7-DIHYDRO-5H-BENZO(7)ANNULENE-3-CARBOXYLIC ACID
Code names
SAR-439859

Resolves to

Compound
UNIITBF1NHY02OCAS2114339-57-8
Targets
P03372ESR1

What you can answer from here — as of June 15, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action
Listed above
7Clinical trialsPhase, status and sponsor resolved per trial
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2+ReferencesStructured and connected to the statements they support
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Which drugs share a target with Amcenestrant, and which of those have an active Phase 3 trial?

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