Reaction: Iptacopan to 1 product
- Reaction
- Reaction type
- O-deethylation
- Direction
- Major circulating metabolite?
- No
- Spontaneous?
- No
- Activity
- inactive
- References
- James AD, Kulmatycki K, Poller B, Romeo AA, Van Lier JJ, Klein K, Pearson D: Absorption, Distribution, Metabolism, and Excretion of [(14)C]iptacopan in Healthy Male Volunteers and in In Vivo and In Vitro Studies. Drug Metab Dispos. 2023 Jul;51(7):873-883. doi: 10.1124/dmd.123.001290. Epub 2023 Jun 12. [Article]
- FDA Approved Drug Products: FABHALTA® (iptacopan) capsules, for oral use [Link]
- Comments
- Not Available
- Enzymes
- Not Available