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Cetermin
go.drugbank.com/drugs/DB32081ExperimentalSynonyms: Tgf-.beta.2 (human), Transforming growth factor-beta 2Piconol
go.drugbank.com/drugs/DB20219ExperimentalPiconol is a small molecule drug. Piconol has a monoisotopic molecular weight of 109.05 Da.
Synonyms: 2-pyridinemethanolSunvozertinib
go.drugbank.com/drugs/DB18925Investigational[A274143] Sunvozertinib was granted accelerated approval in the US on July 2, 2025 for the treatment of locally advanced or metastatic non-small cell lung cancer (NSCLC) with epidermal growth factor … receptor (EGFR) exon 20 insertion mutations.
Synonyms: 2-Propenamide, N-[5-[[4-[[5-chloro-4-fluoro-2-(1-hydroxy-1- methylethyl)phenyl]amino]-2-pyrimidinyl]amino]-2-[(3R)-3-(dimethylamino)-1-pyrrolidinyl]-4-methoxyphenyl]-, N-{5-[(4-{[5-chloro-4-fluoro-2-(1-hydroxy-1-methylethyl)phenyl]amino}pyrimidin-2-yl)amino]-2-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-4-methoxyphenyl}prop-2-enamideCategories: P-glycoprotein inhibitors, Cytochrome P-450 SubstratesMosliciguat
go.drugbank.com/drugs/DB19425InvestigationalMosliciguat is under investigation in clinical trial NCT06635850 (A Phase 2 Study of Mosliciguat in PH-ILD).
Synonyms: (5s)-5-((2-(4-carboxyphenyl)ethyl)(2-(2-((3-chloro-4'-(trifluoromethyl)biphenyl-4-yl)methoxy)phenyl)ethyl)amino)-5,6,7,8-tetrahydroquinoline-2-carboxylic acid, 2-quinolinecarboxylic acid, 5-((2-(4-carboxyphenyl)ethyl)(2-(2-((3-chloro-4'-(trifluoromethyl)(1,1'-biphenyl)-4-yl)methoxy)phenyl)ethyl)amino)-5,6,7,8-tetrahydro-, (5s)-Cyclocreatine
go.drugbank.com/drugs/DB17624ExperimentalSynonyms: 2-imino-1-imidazolidineacetic acid, 1-carboxymethyl-2-imino-imidazolidineCategories: Heterocyclic Compounds, 1-RingCaricotamide
go.drugbank.com/drugs/DB18950InvestigationalCaricotamide is under investigation in clinical trial NCT00746590 (Study of Anti-tumour Effects and Safety of Prolarix™ in Hepatocellular Carcinoma).
Synonyms: 1-(2-amino-2-oxoethyl)-1,4-dihydropyridine-3-carboxamideBHV-5000
go.drugbank.com/drugs/DB17817ExperimentalBHV-5000 is an orally bioavailable, low-trapping, potent N-methyl-D-aspartate (NMDA) receptor antagonist. The active metabolite of BHV-5000 is [lanicemine].[L46446]
Synonyms: (S)-1-(L-valyl)-N_((S)-1-phenyl-2-(pyridin-2-yl)ethyl)pyrrolidine-2-carboxamide fumarateZebularine
go.drugbank.com/drugs/DB03068ExperimentalA chemically stable, cytidine analog that displays anti-tumor properties. It acts as a transition state analog inhibitor of cytidine deaminase by binding to the active site as covalent hydrates.
Categories: Heterocyclic Compounds, 1-RingSynonyms: 1-beta-D-ribofuranosyl-2(1H)-pyrimidinone, 1-beta-D-ribofuranosylpyrimidin-2(1H)-oneMethylisothiazolinone
go.drugbank.com/drugs/DB15884InvestigationalSynonyms: 2-Methyl-3(2H)-isothiazolone, 2-Methyl-3-isothiazoloneCategories: Heterocyclic Compounds, 1-Ring, Compounds used in a research, industrial, or household settingIdroxioleic acid
go.drugbank.com/drugs/DB18213InvestigationalSynonyms: 2-OHOA, (z)-2-hydroxyoctadec-9-enoic acid