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AMG-900
go.drugbank.com/drugs/DB17197ExperimentalSalts: AMG-900 bismesylate dihydrateCategories: Heterocyclic Compounds, 1-RingBisantrene
go.drugbank.com/drugs/DB17247InvestigationalSynonyms: 9,10-anthracenedicarboxaldehyde bis(2-imidazolin-2-ylhydrazone), 9,10-anthracenedicarboxaldehyde, bis((4,5-dihydro-1h-imidazol-2-yl)hydrazone)APPD
go.drugbank.com/drugs/DB18603ExperimentalSynonyms: D-GLYCERO-.ALPHA.-L-TALO-HEPTOFURANURONAMIDE, 5-O-(5-AMINO-5-DEOXY-.BETA., -D-RIBOFURANOSYL)-1,6-DIDEOXY-1-(3,4-DIHYDRO-2,4-DIOXO-1(2H)-PYRIMIDINYL)-6-((4-OXO-4-(((4-(4-(4-(TRIFLUOROMETHOXY)PHENOXY)-1-PIPERIDINYL)PHENYL)METHYL)AMINO)BUTYL)AMINO)-Categories: P-glycoprotein inhibitors, Cytochrome P-450 SubstratesWP-1066
go.drugbank.com/drugs/DB12679InvestigationalWP1066 has been used in trials studying the treatment of Melanoma, Brain Cancer, Solid Tumors, and Central Nervous System Neoplasms.
Synonyms: (E)-3-(6-Bromo-pyridin-2-yl)-2-cyano-N-((S)-1-phenyl-ethyl)-acryl amide, 2-PROPENAMIDE, 3-(6-BROMO-2-PYRIDINYL)-2-CYANO-N-((1S)-1-PHENYLETHYL)-, (2E)-Categories: Heterocyclic Compounds, 2-Ring, Heterocyclic Compounds, 1-RingBrodimoprim
go.drugbank.com/drugs/DB13795ExperimentalSynonyms: 2,4-diamino-5-(4-bromo-3,5-dimethoxybenzyl)pyrimidineCategories: Heterocyclic Compounds, 1-RingCyclocreatine
go.drugbank.com/drugs/DB17624ExperimentalSynonyms: 2-imino-1-imidazolidineacetic acid, 1-carboxymethyl-2-imino-imidazolidineCategories: Heterocyclic Compounds, 1-RingCaricotamide
go.drugbank.com/drugs/DB18950InvestigationalCaricotamide is under investigation in clinical trial NCT00746590 (Study of Anti-tumour Effects and Safety of Prolarix™ in Hepatocellular Carcinoma).
Synonyms: 1-(2-amino-2-oxoethyl)-1,4-dihydropyridine-3-carboxamideAminosalicylic acid
go.drugbank.com/drugs/DB00233ApprovedInvestigationalAn antitubercular agent often administered in association with isoniazid. The sodium salt of the drug is better tolerated than the free acid.
Categories: 4-aminosalicylic acidSynonyms: 4-amino-2-hydroxybenzoic acid, 4-aminosalicylateBHV-5000
go.drugbank.com/drugs/DB17817ExperimentalBHV-5000 is an orally bioavailable, low-trapping, potent N-methyl-D-aspartate (NMDA) receptor antagonist. The active metabolite of BHV-5000 is [lanicemine].[L46446]
Synonyms: (S)-1-(L-valyl)-N_((S)-1-phenyl-2-(pyridin-2-yl)ethyl)pyrrolidine-2-carboxamide fumarateMethylisothiazolinone
go.drugbank.com/drugs/DB15884InvestigationalMixtures: 75% Alcohol WipesCategories: Heterocyclic Compounds, 1-Ring, Compounds used in a research, industrial, or household setting