| DB00067 | Vasopressin | approved | yes | agonistregulator | Details |
| DB00093 | Felypressin | experimental | yes | agonist | Details |
| DB00872 | Conivaptan | approved, investigational | yes | antagonist | Details |
| DB02638 | Terlipressin | approved, investigational | yes | agonist | Details |
| DB00035 | Desmopressin | approved | yes | | Details |
| DB05452 | PH-284 | investigational | unknown | | Details |
| DB06212 | Tolvaptan | approved | no | antagonist | Details |
| DB13929 | Relcovaptan | investigational | unknown | antagonist | Details |
| DB09059 | Atosiban | approved, investigational | unknown | antagonist | Details |
| DB14642 | Lypressin | approved | yes | | Details |
| DB16279 | Pecavaptan | investigational | unknown | antagonist | Details |