| DB00577 | Valaciclovir | approved, investigational | yes | substrate | Details |
| DB00194 | Vidarabine | approved, investigational | yes | inducer | Details |
| DB00249 | Idoxuridine | approved, investigational | unknown | unknown | Details |
| DB00787 | Acyclovir | approved | yes | substrate | Details |
| DB01004 | Ganciclovir | approved, investigational | yes | substrate | Details |
| DB02324 | 5-Iodo-2'-Deoxyuridine-5'-Monophosphate | experimental | unknown | substrate | Details |
| DB02495 | 9-(4-hydroxybutyl)-N2-phenylguanine | experimental | unknown | inhibitor | Details |
| DB02765 | R-9-(2-hydroxypropyl)adenine | experimental | no | ligand | Details |
| DB02500 | 6-(Dihydroxy-Isobutyl)-Thymine | experimental | unknown | substrate | Details |
| DB02921 | (South)-Methanocarba-Thymidine | experimental | unknown | inhibitor | Details |
| DB03804 | 5-Bromothienyldeoxyuridine | experimental | unknown | ligand | Details |
| DB04139 | 6-Hydroxypropylthymine | experimental | unknown | ligand | Details |