GABA-B Receptor Agonists

All categories
Name
GABA-B Receptor Agonists
Accession Number
DBCAT000430
Description

Endogenous compounds and drugs that bind to and activate GABA-B RECEPTORS.

Drugs
DrugDrug Description
Arbaclofen PlacarbilInvestigated for the treatment of spasticity in multiple sclerosis, acute back spasms, and GERD.
BaclofenA GABA-ergic agonist used to manage severe spasticity of cerebral or spinal origin in adult and pediatric patients.
Drugs & Drug Targets
DrugTargetType
Arbaclofen PlacarbilMonocarboxylate transporter 1transporter
Arbaclofen PlacarbilGamma-aminobutyric acid type B receptor subunit 1target
Arbaclofen PlacarbilGamma-aminobutyric acid type B receptor subunit 2target
Arbaclofen PlacarbilGamma-aminobutyric acid receptor subunit gamma-3target
BaclofenGamma-aminobutyric acid type B receptor subunit 1target
BaclofenGamma-aminobutyric acid type B receptor subunit 2target
BaclofenC-X-C chemokine receptor type 4target