Janus Kinase 3, antagonists & inhibitors

Name
Janus Kinase 3, antagonists & inhibitors
Accession Number
DBCAT001910
Description

Not Available

Drugs
DrugDrug Description
TofacitinibA Janus kinase (JAK) inhibitor used to treat rheumatic conditions, such as rheumatoid arthritis and ankylosing spondylitis, and ulcerative colitis.
RitlecitinibA kinase inhibitor used to treat severe alopecia areata in adults and adolescents 12 years and older.
Drugs & Drug Targets
DrugTargetType
TofacitinibNon-receptor tyrosine-protein kinase TYK2target
TofacitinibCytochrome P450 3A4enzyme
TofacitinibCytochrome P450 2C19enzyme
TofacitinibTyrosine-protein kinase JAK2target
TofacitinibTyrosine-protein kinase JAK1target
TofacitinibTyrosine-protein kinase JAK3target
TofacitinibSerum albumincarrier
RitlecitinibTyrosine-protein kinase JAK3target
RitlecitinibTyrosine-protein kinase Tectarget
RitlecitinibTyrosine-protein kinase ITK/TSKtarget
RitlecitinibTyrosine-protein kinase TXKtarget
RitlecitinibTyrosine-protein kinase BTKtarget
RitlecitinibCytoplasmic tyrosine-protein kinase BMXtarget
RitlecitinibCytochrome P450 3A4enzyme
RitlecitinibCytochrome P450 2C8enzyme
RitlecitinibCytochrome P450 1A2enzyme
RitlecitinibCytochrome P450 2C9enzyme
RitlecitinibGlutathione S-transferase A1enzyme
RitlecitinibGlutathione S-transferase A3enzyme
RitlecitinibGlutathione S-transferase Mu 1enzyme
RitlecitinibGlutathione S-transferase Mu 3enzyme
RitlecitinibGlutathione S-transferase Mu 5enzyme
RitlecitinibGlutathione S-transferase Penzyme
RitlecitinibGlutathione S-transferase theta-2enzyme
RitlecitinibMaleylacetoacetate isomeraseenzyme
RitlecitinibMicrosomal glutathione S-transferase 1enzyme
RitlecitinibMicrosomal glutathione S-transferase 2enzyme
RitlecitinibMicrosomal glutathione S-transferase 3enzyme