Human Immunodeficiency Virus Integrase Strand Transfer Inhibitor

Name
Human Immunodeficiency Virus Integrase Strand Transfer Inhibitor
Accession Number
DBCAT003484
Description

Not Available

Drugs
DrugDrug Description
RaltegravirAn antiretroviral agent used for the treatment of HIV infections in conjunction with other antiretrovirals.
DolutegravirAn antiviral agent used for the treatment of HIV-1 infections in combination with other antiretroviral agents.
ElvitegravirAn antiretroviral agent used in combination with other antiretrovirals for the treatment of HIV-1 infection in antiretroviral treatment-experienced adults.
CabotegravirAn HIV-1 integrase inhibitor used for treatment and pre-exposure prophylaxis of HIV-1 infection.
BictegravirAn integrase inhibitor used to treat HIV infections.
Drugs & Drug Targets
DrugTargetType
RaltegravirUDP-glucuronosyltransferase 1-1enzyme
RaltegravirIntegrasetarget
DolutegravirUDP-glucuronosyltransferase 1-1enzyme
DolutegravirCytochrome P450 3A Subfamilyenzyme
DolutegravirIntegrasetarget
DolutegravirSolute carrier family 22 member 2transporter
DolutegravirUDP-glucuronosyltransferase 1-3enzyme
DolutegravirUDP-glucuronosyltransferase 1-9enzyme
DolutegravirATP-binding cassette sub-family G member 2transporter
DolutegravirSolute carrier family 22 member 6transporter
DolutegravirSolute carrier family 22 member 8transporter
DolutegravirP-glycoprotein 1transporter
DolutegravirMultidrug and toxin extrusion protein 1transporter
DolutegravirSerum albumincarrier
Dolutegraviralpha1-acid glycoproteincarrier
ElvitegravirIntegrasetarget
ElvitegravirCytochrome P450 3A4enzyme
ElvitegravirUDP-glucuronosyltransferase 1-1enzyme
CabotegravirSolute carrier family 22 member 6transporter
CabotegravirSolute carrier family 22 member 8transporter
CabotegravirUDP-glucuronosyltransferase 1-1enzyme
CabotegravirUDP-glucuronosyltransferase 1-9enzyme
CabotegravirP-glycoprotein 1transporter
CabotegravirATP-binding cassette sub-family G member 2transporter
CabotegravirSerum albumincarrier
CabotegravirIntegrasetarget
BictegravirReverse transcriptase/RNaseHtarget
BictegravirIntegrasetarget
BictegravirCytochrome P450 3A4enzyme
BictegravirUDP-glucuronosyltransferase 1-1enzyme
BictegravirPOU domain, class 2, transcription factor 2enzyme
BictegravirMultidrug and toxin extrusion protein 1enzyme