Poly (ADP-ribose) polymerase (PARP) inhibitors

Name
Poly (ADP-ribose) polymerase (PARP) inhibitors
Accession Number
DBCAT005743
Description

Not Available

ATC Classification
Drugs
DrugDrug Description
VeliparibNot Available
OlaparibA poly (ADP-ribose) polymerase (PARP) inhibitor used to treat ovarian cancer, breast cancer, pancreatic cancer, and prostate cancer.
TalazoparibA poly-ADP ribose polymerase inhibitor used to treat HER2-, BRCA mutated locally advanced or metastatic breast cancer and HRR gene-mutated metastatic castration-resistant prostate cancer.
NiraparibA poly-ADP ribose polymerase inhibitor used to treat recurrent epithelial ovarian, fallopian tube, or primary peritoneal cancer responding to platinum based chemotherapy.
RucaparibA poly (ADP-ribose) polymerase (PARP) inhibitor used to treat recurrent ovarian and prostate cancers in previously treated adults.
PamiparibPamiparib is under investigation in clinical trial NCT03933761 (Pamiparib in Fusion Positive, Reversion Negative High Grade Serous Ovarian Cancer or Carcinosarcoma With BRCA1/2 Gene Mutations If Progression on Substrate Poly...
AbirateroneAn antiandrogen used in the treatment of metastatic castration-resistant prostate cancer and metastatic high-risk castration-sensitive prostate cancer.
Drugs & Drug Targets
DrugTargetType
VeliparibPoly [ADP-ribose] polymerase 1target
VeliparibPoly [ADP-ribose] polymerase 2target
OlaparibPoly [ADP-ribose] polymerase 1target
OlaparibCytochrome P450 3A4enzyme
OlaparibCytochrome P450 2B6enzyme
OlaparibPoly [ADP-ribose] polymerase 2target
OlaparibProtein mono-ADP-ribosyltransferase PARP3target
OlaparibCytochrome P450 3A5enzyme
OlaparibATP-dependent translocase ABCB1transporter
OlaparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
OlaparibAldo-keto reductase family 1 member C3target
OlaparibUDP-glucuronosyltransferase 1A1enzyme
OlaparibAlbumincarrier
OlaparibAlpha-1-acid glycoprotein 1carrier
TalazoparibPoly [ADP-ribose] polymerase 1target
TalazoparibPoly [ADP-ribose] polymerase 2target
TalazoparibATP-dependent translocase ABCB1transporter
TalazoparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
NiraparibPoly [ADP-ribose] polymerase 1target
NiraparibPoly [ADP-ribose] polymerase 2target
NiraparibCarboxylesteraseenzyme
NiraparibCytochrome P450 1A2enzyme
NiraparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
NiraparibMultidrug and toxin extrusion protein 1transporter
NiraparibMultidrug and toxin extrusion protein 2transporter
NiraparibATP-dependent translocase ABCB1transporter
NiraparibAlbumincarrier
RucaparibPoly [ADP-ribose] polymerase 1target
RucaparibPoly [ADP-ribose] polymerase 2target
RucaparibProtein mono-ADP-ribosyltransferase PARP3target
RucaparibCytochrome P450 2D6enzyme
RucaparibCytochrome P450 1A2enzyme
RucaparibCytochrome P450 3A4enzyme
RucaparibATP-dependent translocase ABCB1transporter
RucaparibBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
RucaparibMultidrug and toxin extrusion protein 1transporter
RucaparibMultidrug and toxin extrusion protein 2transporter
RucaparibSolute carrier family 22 member 1transporter
RucaparibATP-binding cassette sub-family C member 4transporter
RucaparibSolute carrier organic anion transporter family member 1B1transporter
RucaparibSolute carrier organic anion transporter family member 1B3transporter
RucaparibSolute carrier family 22 member 6transporter
RucaparibOrganic anion transporter 3transporter
RucaparibCytochrome P450 3A5enzyme
RucaparibCytochrome P450 3A7enzyme
RucaparibCytochrome P450 3A43enzyme
RucaparibCytochrome P450 2C19enzyme
RucaparibCytochrome P450 2C9enzyme
RucaparibCytochrome P450 2C8enzyme
RucaparibUDP-glucuronosyltransferase 1A1enzyme
AbirateroneSteroid 17-alpha-hydroxylase/17,20 lyasetarget
AbirateroneAlbumincarrier
AbirateroneAlpha-1-acid glycoprotein 1carrier
AbirateroneCytochrome P450 3A4enzyme
AbirateroneSulfotransferase 2A1enzyme
AbirateroneMultidrug resistance-associated protein 1transporter
AbirateroneCytochrome P450 2D6enzyme
AbirateroneCytochrome P450 2C8enzyme
AbirateroneCytochrome P450 1A2enzyme
AbirateroneCytochrome P450 2C19enzyme
AbirateroneCytochrome P450 2C9enzyme
AbirateroneCytochrome P450 3A5enzyme
AbirateroneSolute carrier organic anion transporter family member 1B1transporter