Epitestosterone

DB07768ExperimentalSmall molecule

Epitestosterone is the 17-alpha isomer of testosterone, derived from pregnenolone via the delta5-steroid pathway, and via 5-androstene-3-beta,17-alpha-diol. Epitestosterone acts as an antiandrogen in various target tissues. The ratio between testosterone/epitestosterone... The ratio between testosterone/epitestosterone is used to monitor anabolic drug abuse.

Formula / weight: C₁₉H₂₈O₂ · 288.4244 g/mol (avg)
Also known as: 17-alpha-Testosterone · 17-Epitestosterone · 17alpha-cis-Testosterone · cis-Testosterone · Isotestosterone
Code names: NSC-26499

Resolves to

Compound

UNII48L726977ZCAS481-30-1ChEMBLCHEMBL196228ChEBI42534PubChem10204

Structure

InChIKeyMUMGGOZAMZWBJJ-KZYORJDKSA-NSMILES[H][C@@]1(O)CC[C@@]2([H])[C@]3([H])CCC4=CC(=O)CC[C@]4(C)[C@@]3([H])CC[C@]12C

Targets

Q04828AKR1C1P52895AKR1C2

What you can answer from here — as of June 12, 2020

2Protein targetsEach mapped to UniProt, with action and pharmacological action

Listed above

62Drug interactionsStructured to mechanism, not free text

2+ReferencesStructured and connected to the statements they support

Which drugs share a target with Epitestosterone, and which of those have an active Phase 3 trial?

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