Tilidine

DB13787InvestigationalSmall molecule

Tilidine is a synthetic opioid indicated in the treatment of severe pain. A medication used to treat severe pain.

Mechanism: Pharmacologically active on Mu-type opioid receptor
Curator reviewed
Formula / weight: C₁₇H₂₃NO₂ · 273.376 g/mol (avg)
Also known as: Tilidate
Code names: DEA No. 9750

Resolves to

Compound

Clinical / RWD

Structure

InChIKeyWDEFBBTXULIOBB-WBVHZDCISA-NSMILESCCOC(=O)[C@@]1(CCC=C[C@H]1N(C)C)C1=CC=CC=C1

Targets

Transporters

What you can answer from here — as of September 14, 2026

1Protein targetEach mapped to UniProt, with action and pharmacological action

Listed above

1TransporterSubstrate / inhibitor direction, not just membership

Listed above

919Drug interactionsStructured to mechanism, not free text

1Structured indicationCondition, population, route and combination as fields, not prose

6ContraindicationsEach with its own population and attribute set

94Marketed productsAcross every region we cover

2ATC codesIncluding every combination product, plus 25 drug categories

10+ReferencesStructured and connected to the statements they support

Which drugs share a target with Tilidine, and which of those have an active Phase 3 trial?

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