TPMPA

DB16754ExperimentalSmall molecule

TPMPA ((1,2,5,6-tetrahydropyridine-4-yl)methylphosphinic acid) is a selective antagonist of GABAC receptors (also known as GABA-ρ or GABAA-ρ receptors). GABAC receptors are found primarily in the retina, although they may be present... GABAC receptors are found primarily in the retina, although they may be present in other tissues, including the hippocampus, spinal cord, superior colliculus, pituitary and the gut.

Chemical structure of TPMPA
Formula / weight
C6H12NO2P · 161.141 g/mol (avg)

Resolves to

Structure
InChIKeyMFUKVPOVVKKLRQ-UHFFFAOYSA-NSMILESCP(O)(=O)C1=CCNCC1

What you can answer from here — as of April 02, 2025

3Protein targetsEach mapped to UniProt, with action and pharmacological action
Listed above
7+ReferencesStructured and connected to the statements they support
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