Feloprentan

DB20151ExperimentalSmall molecule

Feloprentan is a small molecule drug. The usage of the INN stem '-entan' in the name indicates that Feloprentan is a endothelin receptor antagonist. Feloprentan has a monoisotopic molecular weight...

Formula / weight: C₃₁H₃₂N₂O₆ · 528.605 g/mol (avg)
Code names: LU-302872

Resolves to

Compound

UNII6RW6H4951ZCAS204267-34-5ChEMBLCHEMBL316735ChEBI748437PubChem9893800

Structure

InChIKeyCLSJNXXMIVKULC-MUUNZHRXSA-NSMILESCOC1=CC=C(CCOC([C@H](OC2=NC(C)=CC(C)=N2)C(O)=O)(C2=CC=CC=C2)C2=CC=CC=C2)C=C1OC

Targets

P24530EDNRBP25101EDNRA

What you can answer from here — as of September 23, 2026

2Protein targetsEach mapped to UniProt, with action and pharmacological action

Listed above

6+ReferencesStructured and connected to the statements they support

Which drugs share a target with Feloprentan, and which of those have an active Phase 3 trial?

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