Ledaborbactam

DB21457ExperimentalSmall molecule

Ledaborbactam is a small molecule drug. The usage of the INN stem '-bactam' in the name indicates that Ledaborbactam is a ẞ-lactamase inhibitor. Ledaborbactam has a monoisotopic molecular weight of...

Mechanism: Pharmacologically active on Beta-lactamase, Beta-lactamase CTX-M, and OXA-48 carbapenemase
Curator reviewed
Formula / weight: C₁₂H₁₄BNO₅ · 263.06 g/mol (avg)
Code names: VNRX-5236 · VNRX-7145 ACID · VNRX-7145 ACTIVE METABOLITE

Resolves to

Compound

UNIIG2WGD69BLICAS1842397-36-7ChEMBLCHEMBL5093566ChEBI758608PubChem138455079

Structure

InChIKeyQAGGLFCWUVSERJ-VIFPVBQESA-NSMILESCCC(=O)N[C@H]1CC2=C(OB1O)C(=CC=C2)C(O)=O

Targets

P00811ampCA0A023W3H0OXA-48Q9F663KPC-2

What you can answer from here — as of September 23, 2026

4Protein targetsEach mapped to UniProt, with action and pharmacological action

Listed above

11+ReferencesStructured and connected to the statements they support

Which drugs share a target with Ledaborbactam, and which of those have an active Phase 3 trial?

Answer this in Biopharma OS Sign in to your account

Create a free account or log in to explore the full data card.

Create Account