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Purvalanol A
go.drugbank.com/drugs/DB04751ExperimentalSynonyms: 2-(1R-Isopropyl-2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine, Purvalanol ACategories: Heterocyclic Compounds, 2-RingTryptamine
go.drugbank.com/drugs/DB08653InvestigationalSynonyms: 2-(3-indolyl)ethylamine, 3-(2-Aminoethyl)indoleCategories: Heterocyclic Compounds, 2-Ring, Monoamine Oxidase A Inhibitors for interaction with Monoamine Oxidase A substratesAtilotrelvir
go.drugbank.com/drugs/DB19439InvestigationalAtilotrelvir is under investigation in clinical trial NCT05041907 (Finding Treatments for COVID-19: A Trial of Antiviral Pharmacodynamics in Early Symptomatic COVID-19 (PLATCOV)).
Synonyms: Spiro[2-azabicyclo[2.2.1]heptane-5,1′-cyclopropane]-3-carboxamide, N-[(1S)-1-cyano-2-[(3S)-2-oxo-3-pyrrolidinyl]ethyl]-2-[(2S)-3,3-dimethyl-1-oxo-2-[(2,2,2-trifluoroacetyl)amino]butyl]-, (1S,3S,4R)-, (1R,4S,6S)-N-{(1S)-1-ciano-2-[(3S)-2-oxopirrolidin-3-il]etil}-5-[(2S)-3,3-dimetil-2-(2,2,2-trifluoroacetamido)butanoil]-5-azaespiro[biciclo[2.2.1]heptano-2,1'-ciclopropano]-6-carboxamidaFlutafuranol F-18
go.drugbank.com/drugs/DB18825ExperimentalSynonyms: 2-(2-(18f)fluoro-6-(methylamino)pyridin-3-yl)-1-benzofuran-5-ol, 5-benzofuranol, 2-(2-(fluoro-18f)-6-(methylamino)-3-pyridinyl)-PXS-4728A free base
go.drugbank.com/drugs/DB19177InvestigationalPXS-4728A free base is under investigation in clinical trial NCT05904717 (Effect of PXS-4728A on Microglia Activation in Participants With Isolated Rapid Eye Movement Sleep Behaviour Disorder).
Synonyms: Benzamide, 4-(((2e)-2-(aminomethyl)-3-fluoro-2-propen-1-yl)oxy)-n-(1,1-dimethylethyl)-CRA_16847
go.drugbank.com/drugs/DB02063ExperimentalSynonyms: 2-(3-{5-[AMINO(IMINIO)METHYL]-1H-BENZIMIDAZOL-2-YL}-5-BROMO-4-OXIDOPHENYL)SUCCINATEN-acetyl-D-glucosamine-6-phosphate
go.drugbank.com/drugs/DB03951ExperimentalSynonyms: 2-acetamido-2-deoxy-6-O-phosphono-D-glucopyranose, N-acetyl-D-glucosamine-6-phosphateEsmirtazapine
go.drugbank.com/drugs/DB06678InvestigationalThis includes inverse agonist activity of H1 and 5-HT2 receptors and antagonism of α2-adrenergic receptors. … Esmirtazapine is the (S)-(+)-enantiomer of mirtazapine and possesses similar overall pharmacology.
Synonyms: (S)-1,2,3,4,10,14b-hexahydro-2-methylpyrazino(2,1-a)pyrido(2,3-c)(2)benzazepineCategories: Adrenergic alpha-2 Receptor Antagonists, Cytochrome P-450 SubstratesN-BENZYLOXYCARBONYL-ALA-PRO-3-AMINO-4-PHENYL-BUTAN-2-OL
go.drugbank.com/drugs/DB06886ExperimentalSynonyms: N-BENZYLOXYCARBONYL-ALA-PRO-3-AMINO-4-PHENYL-BUTAN-2-OL4-(2-Oxo-Hexahydro-Thieno[3,4-D]Imidazol-4-Yl)-Butyricacid
go.drugbank.com/drugs/DB02674ExperimentalSynonyms: 4-(2-Oxo-Hexahydro-Thieno[3,4-D]Imidazol-4-Yl)-Butyricacid