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Elraglusib
go.drugbank.com/drugs/DB16047InvestigationalElraglusib is under investigation in clinical trial NCT04218071 (Actuate 1901: 9-ING-41 in Myelofibrosis).
Synonyms: 1H-Pyrrole-2,5-dione, 3-(5-fluoro-3-benzofuranyl)-4-(5-methyl-5H-1,3-dioxolo(4,5-F)indol-7-yl)-, 3-(5-Fluoro-benzofuran-3-yl)-4-(5-methyl-5H-(1,3)dioxolo(4,5-F)indol-7-yl)-pyrrole-2,5-dioneSaruparib
go.drugbank.com/drugs/DB18982Investigational(IHC 0, 1+, 2+/ ISH Non-amplified), BRCA1, BRCA2, or Palb2m Advanced Breast Cancer). … Saruparib is under investigation in clinical trial NCT06380751 (Saruparib (AZD5305) Plus Camizestrant Compared With CDK4/6 Inhibitor Plus Endocrine Therapy or Plus Camizestrant in Hr-positive, Her2-negative
Categories: Heterocyclic Compounds, 1-Ring, Heterocyclic Compounds, 2-RingSynonyms: 2-Pyridinecarboxamide, 5-[4-[(7-ethyl-5,6-dihydro-6-oxo-1,5-naphthyridin-3-yl)methyl]-1-piperazinyl]-N-methyl-, 5-{4-[(7-ethyl-5,6-dihydro-6-oxo-1,5-naphthyridin-3- yl)methyl]piperazin-1-yl}-N-methylpyridine-2- carboxamideVocacapsaicin
go.drugbank.com/drugs/DB17071InvestigationalSynonyms: 1-piperidinecarboxylic acid, 2-((methylamino)methyl)-, 2-methoxy-4-((((6e)-8-methyl-1-oxo-6-nonen-1-yl)amino)methyl) phenyl ester, 2-methoxy-4-(((6e)-8-methylnon-6-enamido)methyl)phenyl (2rs)-2-((methylamino)methyl)piperidine-1-carboxylateMonepantel
go.drugbank.com/drugs/DB18755InvestigationalSynonyms: Benzamide, n-((1s)-1-cyano-2-(5-cyano-2-(trifluoromethyl)phenoxy)-1-methylethyl)-4-((trifluoromethyl)thio)-, N-(2-cyano-1-((2s)-5-cyano-2-(trifluoromethyl)phenoxy)propan-2-yl)-4-(trifluoromethylsulfanyl)benzamideMePPEP C-11
go.drugbank.com/drugs/DB19280ExperimentalSynonyms: (3r,5r)-5-(3-11c-methoxy-phenyl)-3-((r)-1-phenyl-ethylamino)-1-(4-trifluoromethyl-phenyl)-pyrrolidin-2-one, 2-pyrrolidinone, 5-(3-(methoxy-11c)phenyl)-3-(((1r)-1-phenylethyl)amino)-1-(4-(trifluoromethyl)phenyl)-, (3r,5r)-Vamifeport
go.drugbank.com/drugs/DB17692InvestigationalVamifeport is being investigated for the treatment of beta-thalassemia.
Synonyms: 2-(2-((2-(1h-benzimidazol-2-yl)ethyl)amino)ethyl)-n-((3-fluoropyridin-2-yl)methyl)-1,3-oxazole-4-carboxamide, 4-oxazolecarboxamide, 2-(2-((2-(1h-benzimidazol-2-yl)ethyl)amino)ethyl)-n-((3-fluoro-2-pyridinyl)methyl)-Categories: Heterocyclic Compounds, 1-Ring, Heterocyclic Compounds, 2-RingLB-102
go.drugbank.com/drugs/DB19214InvestigationalLB-102 is under investigation in clinical trial NCT06179108 (Randomized, Double-blinded, Placebo-controlled, Evaluating the Treatment With LB-102 in Patients With Acute Schizophrenia).
Synonyms: Benzamide, n-((1-ethyl-2-pyrrolidinyl)methyl)-5-(ethylsulfonyl)-2-methoxy-4-(methylamino)-, N'-methylamisulprideGosogliptin
go.drugbank.com/drugs/DB08382InvestigationalGosogliptin has been used in trials studying the treatment of Renal Insufficiency, Chronic.
Categories: Heterocyclic Compounds, 1-Ring, Diabetes Mellitus, Type 2, drug therapySynonyms: 2-(4-{(3S,5S)-5-[(3,3-difluoropyrrolidin-1-yl)carbonyl]pyrrolidin-3-yl}piperazin-1-yl)pyrimidineSulfathiourea
go.drugbank.com/drugs/DB13699ExperimentalSynonyms: 4-amino-N-(aminothioxomethyl)benzenesulfonamide, 1-sulfanilyl-2-thiourea2-(p-Tolyl)ethyl nicotinate
go.drugbank.com/drugs/DB16617InvestigationalSynonyms: 3-pyridinecarboxylic acid, 2-(4-methylphenyl)ethyl ester , 2-(p-Tolyl)ethyl nicotinate