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Inlexisertib
go.drugbank.com/drugs/DB21713InvestigationalInlexisertib is a small molecule drug. The usage of the INN stem '-sertib' in the name indicates that Inlexisertib is a serine/threonine kinase inhibitor. … Inlexisertib has a monoisotopic molecular weight of 535.29 Da.
Lecufexor
go.drugbank.com/drugs/DB21714ExperimentalLecufexor is a small molecule drug. Lecufexor has a monoisotopic molecular weight of 618.05 Da.
Matsupexole
go.drugbank.com/drugs/DB21715ExperimentalMatsupexole is a small molecule drug. Matsupexole has a monoisotopic molecular weight of 446.25 Da.
Balinatunfib
go.drugbank.com/drugs/DB21728InvestigationalBalinatunfib is a small molecule drug. Balinatunfib has a monoisotopic molecular weight of 502.19 Da.
Cenacitinib
go.drugbank.com/drugs/DB21735InvestigationalCenacitinib is a small molecule drug. The usage of the INN stem '-citinib' in the name indicates that Cenacitinib is a Janus kinase inhibitor. … Cenacitinib has a monoisotopic molecular weight of 431.15 Da.
Certociclib
go.drugbank.com/drugs/DB21736InvestigationalCertociclib is a small molecule drug. Certociclib is under investigation in clinical trial NCT05252416 ((VELA) Study of BLU-222 in Advanced Solid Tumors). … Certociclib has a monoisotopic molecular weight of 365.14 Da.
Rogocekib
go.drugbank.com/drugs/DB21739InvestigationalRogocekib is a small molecule drug. Rogocekib has a monoisotopic molecular weight of 408.15 Da.
Tersolisib
go.drugbank.com/drugs/DB21752InvestigationalSTX-478 is under investigation in clinical trail NCT05768139 (First-in-Human Study of STX-478 as Monotherapy and in Combination With Other Antineoplastic Agents in Participants With Advanced Solid Tumors
Daraxonrasib
go.drugbank.com/drugs/DB22308ApprovedInvestigationalRAS variants rather than a single mutation. … [L64039] It is a RAS(ON) tri-complex inhibitor that binds cyclophilin A and targets the active, GTP-bound ("ON") state of RAS, suppressing signaling of both wild-type and mutant RAS across the most common
Categories: P-glycoprotein inhibitors, P-glycoprotein substrates