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Neflamapimod
go.drugbank.com/drugs/DB07138InvestigationalNeflamapimod has been used in trials studying the treatment of Alzheimer's Disease and Mild Cognitive Impairment.
Categories: Heterocyclic Compounds, 1-RingCA-074 methyl ester
go.drugbank.com/drugs/DB07223ExperimentalCA-074 methyl ester (CA-074Me) is a cell-permeable cathepsin B inhibitor. It is converted by cellular esterases to CA-074.[A258234,A258239]
Synonyms: (S)-methyl 1-((2S,3S)-3-methyl-2-((2S,3S)-3-(propylcarbamoyl)oxirane-2-carboxamido)pentanoyl)pyrrolidine-2-carboxylate, Methyl N-({(2s,3s)-3-[(propylamino)carbonyl]oxiran-2-Yl}carbonyl)-L-isoleucyl-L-prolinateCategories: Cathepsin B, antagonists & inhibitorsVeliparib
go.drugbank.com/drugs/DB07232InvestigationalSynonyms: 2-[(R)-2-methylpyrrolidin-2-yl]-1H-benzimadazole-4-carboxamide, (2R)-2-(7-carbamoyl-1H-benzimidazol-2-yl)-2-methylpyrrolidiniumCategories: Heterocyclic Compounds, 2-RingBMS-564929
go.drugbank.com/drugs/DB07286ExperimentalBMS-564929 is an investigational therapeutic agent built to be a selective androgen receptor modulator (SARM).
Categories: Heterocyclic Compounds, 1-Ring1-(adamantan-1-yl)-2-(1H-imidazol-1-yl)ethanone
go.drugbank.com/drugs/DB07342ExperimentalSynonyms: 1-(adamantan-1-yl)-2-(1H-imidazol-1-yl)ethanoneCategories: Heterocyclic Compounds, 1-Ring, Heme Oxygenase-1, antagonists & inhibitorsAnisomycin
go.drugbank.com/drugs/DB07374ExperimentalAnisomycin (sometimes known as flagecidin), is an antibiotic retrieved from the bacteria Streptomyces griseolus. This drug acts to inhibit bacterial protein and DNA synthesis.
Categories: Heterocyclic Compounds, 1-Ring2-[3-(5-Mercapto-[1,3,4]thiadiazol-2-yl)-ureido]-N-methyl-3-phenyl-propionamide
go.drugbank.com/drugs/DB07390ExperimentalCategories: Heterocyclic Compounds, 1-RingS-23
go.drugbank.com/drugs/DB07419ExperimentalAn androgen receptor modulator.
Synonyms: (2S)-3-(4-Chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide, (+)-S-23Categories: Heterocyclic Compounds, 2-Ring