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Cafedrine
go.drugbank.com/drugs/DB12926InvestigationalCafedrine is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP1A2 SubstratesTheodrenaline
go.drugbank.com/drugs/DB12927InvestigationalTheodrenaline is under investigation in clinical trial NCT01311414 (Effect of Cafedrine/Theodrenaline and Urapidil on Cerebral Oxygenation).
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP1A2 SubstratesTirilazad
go.drugbank.com/drugs/DB13050InvestigationalTirilazad has been used in trials studying the treatment of Spinal Cord Injury.
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP3A SubstratesNorflurane
go.drugbank.com/drugs/DB13116ApprovedInvestigationalWithdrawnNorflurane is under investigation in clinical trial NCT01673061 (Vapocoolant Spray for Numbing Small Boils Before Incision and Drainage).
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP2E1 SubstratesArtemisinin
go.drugbank.com/drugs/DB13132InvestigationalArtemisinin has been used in trials studying the treatment of Schizophrenia, Malaria, Falciparum, and Plasmodium Falciparum.
Categories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP2B6 InducersEsculin
go.drugbank.com/drugs/DB13155ApprovedVitamin C2 is generally considered a bioflavanoid, related to vitamin P esculin is a glucoside that naturally occurs in the horse chestnut (Aesculus hippocastanum), California Buckeye (Aesculus californica
Synonyms: esculetin 6-β-D-glucoside, 6-(beta-D-Glucopyranosyloxy)-7-hydroxy-cumarinGuaiazulen
go.drugbank.com/drugs/DB13329InvestigationalCategories: Cytochrome P-450 CYP1A2 Inhibitors, Cytochrome P-450 Enzyme InhibitorsFlurithromycin
go.drugbank.com/drugs/DB13338ExperimentalCategories: Cytochrome P-450 CYP3A Inhibitors, Cytochrome P-450 CYP3A4 InhibitorsEsatenolol
go.drugbank.com/drugs/DB13443ExperimentalEsatenolol is a beta blocker.
Synonyms: 2-(p-((2S)-2-hydroxy-3-(isopropylamino)propoxy)phenyl)acetamideCategories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP2D6 SubstratesProxyphylline
go.drugbank.com/drugs/DB13449ExperimentalCategories: Cytochrome P-450 Substrates, Cytochrome P-450 CYP1A2 Substrates