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Displaying results 1 - 10 of 12 in total
  1. Drug

    Octreotide

    go.drugbank.com/drugs/DB00104
    ApprovedInvestigational

    [L14513] In the past, octreotide has been administered solely by injection. … [L14501] Octreotide is a long-acting drug with pharmacologic activities that mimic those of the natural hormone, somatostatin, which inhibits the secretion of growth hormone.

    Synonyms: Octreotide, OctreotidaSalts: Octreotide acetate, Octreotide pamoate
  2. Drug

    99mTc-HYNIC (Tyr3)-octreotide

    go.drugbank.com/drugs/DB17161
    Experimental

    Synonyms: 99mTc-HYNIC (Tyr3)-octreotide, 99mTc-HYNIC-[D-Phe1,Tyr3-Octreotide]Salts: 99mTc-HYNIC (Tyr3)-octreotide trifluoroacetate
  3. Drug

    Edotreotide gallium Ga-68

    go.drugbank.com/drugs/DB15494
    Approved

    Edotreotide gallium Ga-68 is an 8 amino acid peptide bound to the chelator 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid (DOTA). Edotreotide gallium Ga-68 is indicated for localizing somatostatin receptor positive neuroendocri...

    Synonyms: Gallium-68 (DOTA0-Phel-Tyr3)octreotide
  4. Drug

    Dotatoc gallium Ga-68

    go.drugbank.com/drugs/DB18190
    Investigational

    Synonyms: Dota-nal3-octreotide Ga-68
  5. Drug

    Edotreotide yttrium Y-90

    go.drugbank.com/drugs/DB17160
    Investigational

    Synonyms: 90y-dota-tyr3-octreotide, Y-90 dota-tyr(3)-octreotide
  6. Drug

    Pasireotide

    go.drugbank.com/drugs/DB06663
    ApprovedInvestigational

    Pasireotide is a synthetic long-acting cyclic hexapeptide with somatostatin-like activity. It is marketed as a diaspartate salt called Signifor, which is used in the treatment of Cushing's disease.

    Salts: Pasireotide acetate
  7. Drug

    Lutetium Lu177 Edotreotide

    go.drugbank.com/drugs/DB17278
    Investigational

    Synonyms: Lutetium Lu-177 dota-tyr3-octreotide
  8. Drug

    Lutetium Lu 177 dotatate

    go.drugbank.com/drugs/DB13985
    ApprovedInvestigational

    survival compared to patients receiving octreotide alone and there was evidence of an overall survival benefit [A31697]. … Compared to the alternative somatostatin analogue DOTA-Tyr3-octreotide (dotatoc), Lutetium Lu 177 dotatate displays higher uptake of radioactivity in tumors and better residence times [A31696].

    Synonyms: 177Lu-Octreotate, 177 Lu-DOTA-octreotate
  9. Indication

    Metastatic Carcinoid Tumors

    go.drugbank.com/conditions/DBCOND0080526
    Drugs: Octreotide
  10. Drug

    Copper oxodotreotide Cu-64

    go.drugbank.com/drugs/DB15873
    Approved

    Further, PET using Copper Cu 64 dotatate has been found to perform better than the current gold standard of single-photon emission computed tomography (SPECT) using 111In-DTPA-octreotide.