| DB03185 | 1-Beta-Ribofuranosyl-1,3-Diazepinone | experimental | unknown | | Details |
| DB00441 | Gemcitabine | approved | unknown | substrate | Details |
| DB00987 | Cytarabine | approved, investigational | unknown | substrate | Details |
| DB00928 | Azacitidine | approved, investigational | unknown | substrate | Details |
| DB01101 | Capecitabine | approved, investigational | unknown | substrate | Details |
| DB03185 | 1-Beta-Ribofuranosyl-1,3-Diazepinone | experimental | unknown | ligand | Details |
| DB15694 | Cedazuridine | approved, investigational | yes | inhibitor | Details |
| DB01262 | Decitabine | approved, investigational | no | substrate | Details |