Diterpenes

Name
Diterpenes
Accession Number
DBCAT000381
Description

Twenty-carbon compounds derived from MEVALONIC ACID or deoxyxylulose phosphate.

Drugs
DrugDrug Description
PhylloquinoneA fat soluble vitamin used to treat hemorrhagic conditions in infants and coumarin overdoses.
ColforsinPotent activator of the adenylate cyclase system and the biosynthesis of cyclic AMP. From the plant Coleus forskohlii. Has antihypertensive, positive inotropic, platelet aggregation inhibitory, and smooth muscle relaxant activities;...
Vitamin AA vitamin important for retinal function that is used clinically to correct vitamin A deficiency.
MenadioneThe primary known function of vitamin K is to assist in the normal clotting of blood, but it may also play a role in normal bone calcification.
AlitretinoinA vitamin A derivative used to treat Kaposi's sarcoma and used off label to treat chronic hand eczema and psoriasis.
TretinoinA vitamin A derivative used to treat acne vulgaris and certain types of promyelocytic leukemia, as well as various skin conditions in over-the-counter medications.
PaclitaxelA taxoid chemotherapeutic agent used as first-line and subsequent therapy for the treatment of advanced carcinoma of the ovary, and other various cancers including breast and lung cancer.
DocetaxelA taxoid antineoplastic agent used in the treatment of various cancers, such as locally advanced or metastatic breast cancer, metastatic prostate cancer, gastric adenocarcinoma, and head and neck cancer.
CarboxyatractylosideNot Available
4-OxoretinolNot Available
Anhydrovitamin ANot Available
N-EthylretinamideN-Ethylretinamide is the ethylamide of all-trans B-retinoic acid.
EcabetFor the treatment of reflux oesophagitis and peptic ulcer disease.
Paclitaxel docosahexaenoic acidInvestigated for use/treatment in breast cancer, colorectal cancer, gastric cancer, kidney cancer, lung cancer, pancreatic cancer, prostate cancer, and skin cancer.
AI-850Investigated for use/treatment in breast cancer and solid tumors.
Paclitaxel trevatideInvestigated for use/treatment in brain cancer.
Ginkgolide AGinkgolide A is a highly active PAF antagonist cage molecule that is isolated from the leaves of the Ginkgo biloba tree. Shows potential in a wide variety of inflammatory and...
ginkgolide-CNot Available
ginkgolide-JNot Available
CabazitaxelAn antineoplastic agent used in combination with corticosteroids to treat metastatic castration-resistant prostate cancer in patients previously treated with a docetaxel-containing treatment regimen.
Gibberellic acidNot Available
Gibberellin A4Not Available
OrtataxelOrtataxel has been used in trials studying the treatment of Lymphoma, Lung Cancer, Glioblastoma, and Kidney Cancer.
TesetaxelTesetaxel has been used in trials studying the treatment of Cancer, Melanoma, Prostate Cancer, Gastric Carcinoma, and Advanced Melanoma, among others.
MenatetrenoneA form of vitamin K2 which is used in the treatment of osteoporosis to stimulate osteogenesis.
Salvinorin ASalvinorin A has been investigated for the basic science of Pharmaceutical Preparations.
MilataxelMilataxel has been used in trials studying the treatment of Mesothelioma.
SteviolbiosideSteviolbioside has been used in trials studying the treatment of HIV-1 Infection.
BMS-188797BMS-188797 has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.
BMS-184476BMS-184476 has been used in trials studying the treatment of Unspecified Adult Solid Tumor, Protocol Specific.
LarotaxelLarotaxel has been used in trials studying the treatment of Cancer, Metastases, Breast Cancer, Breast Neoplasms, and Pancreatic Neoplasms, among others.
Menaquinone 7Menaquinone 7 is under investigation in clinical trial NCT00402974 (The Effect of Vitamin K Supplementation on Osteocalcin Carboxylation in Healthy Children).
MotretinideNot Annotated
Paclitaxel poliglumexNot Annotated
13-cis-12-(3'-Carboxyphenyl)retinoic acidNot Annotated
Menadiol diphosphateNot Annotated
Menaquinone 6Menaquinone 6 is under investigation in clinical trial NCT01194778 (Comparison of Efficacy of Different Dosages Vitamin K2).
Rebaudioside ARebaudioside A is under investigation in clinical trial NCT03510624 (Acute Effect of Rebaudioside A on Glucose Excursion During an Oral Glucose Tolerance Test in Type 2 Diabetes Mellitus).
MenaquinoneMenaquinone is under investigation in clinical trial NCT01533441 (Vitamin K2 Intervention in Patients With Vitamin K Antagonists).
SimotaxelSimotaxel is under investigation in clinical trial NCT00088647 (Study Evaluating MST-997 in Advanced Malignant Solid Tumors).
Menadione bisulfiteNot Annotated
IsosteviolNot Annotated
SteviosideNot Annotated
Tanshinone INot Annotated
Phorbol 12-myristate 13-acetate diesterPhorbol 12-myristate 13-acetate diester is an inducer of neutrophil extracellular traps (NETs).
TPI-287Not Annotated
Paclitaxel ceribateNot Available
TranscrocetinateInvestigated for use/treatment in cancer/tumors (unspecified), hemorrhage, hypoxia, respiratory failure, and strokes.
AphidicolinAphidicolin is an antimitotic and antiviral metabolite of the mould Cephalosporium aphidicola. It inhibits DNA polymerase alpha and blocks DNA replication.[A259157, A259162]
ANG1005Not Annotated
OridoninOridonin is under investigation in clinical trial NCT05130892 (Effect of Inflammasome Inhibitor on Hscrp in Patients After PCI).
Drugs & Drug Targets
DrugTargetType
PhylloquinoneVitamin K-dependent gamma-carboxylasetarget
PhylloquinoneOsteocalcintarget
PhylloquinoneCytochrome P450 4F2enzyme
PhylloquinoneUbiA prenyltransferase domain-containing protein 1enzyme
PhylloquinoneVitamin K epoxide reductase complex subunit 1enzyme
ColforsinATP-dependent translocase ABCB1transporter
ColforsinAdenylate cyclase type 2target
ColforsinGuanine nucleotide-binding protein G(s) subunit alpha isoforms shorttarget
ColforsinAdenylate cyclase type 5target
ColforsinCystic fibrosis transmembrane conductance regulatortarget
ColforsinAdenylate cyclasetarget
ColforsinCalcium-activated potassium channeltarget
ColforsinCREB-binding proteintarget
ColforsinExtracellular signal-regulated kinase (ERK)target
ColforsinMucin-2target
ColforsinPlasminogen activator inhibitor 1target
Vitamin ARetinol dehydrogenase 12target
Vitamin ARetinol dehydrogenase 5target
Vitamin ARetinol dehydrogenase 13target
Vitamin ARetinol-binding protein 5carrier
Vitamin ARetinoid-binding protein 7carrier
Vitamin ARetinol-binding protein 4carrier
Vitamin ARetinol-binding protein 2carrier
Vitamin ARetinal dehydrogenase 2target
Vitamin AAldehyde dehydrogenase 1A1target
Vitamin ALecithin retinol acyltransferasetarget
Vitamin AShort-chain dehydrogenase/reductase 3target
Vitamin ARetinaldehyde dehydrogenase 3target
Vitamin AAll-trans-retinol 13,14-reductasetarget
Vitamin ARetinol dehydrogenase 11target
Vitamin ADehydrogenase/reductase SDR family member 4target
Vitamin ARetinol dehydrogenase 14target
Vitamin ARetinol dehydrogenase 8target
Vitamin ACytochrome P450 26A1enzyme
Vitamin AApolipoprotein Dtarget
Vitamin AProstaglandin-H2 D-isomerasetarget
Vitamin AAlbumincarrier
Vitamin ARetinaldehyde-binding protein 1carrier
Vitamin ARetinol-binding protein 3carrier
Vitamin ARetinol-binding protein 1carrier
Vitamin AReceptor for retinol uptake STRA6transporter
Vitamin ARetinoic acid receptor RXR-gammatarget
MenadioneProthrombintarget
MenadioneVitamin K epoxide reductase complex subunit 1target
MenadioneCoagulation factor IXtarget
MenadioneVitamin K-dependent gamma-carboxylasetarget
MenadioneVitamin K-dependent protein Ctarget
MenadioneVitamin K-dependent protein Starget
MenadioneNAD(P)H dehydrogenase [quinone] 1target
MenadioneRibosyldihydronicotinamide dehydrogenase [quinone]target
MenadioneVitamin K epoxide reductase complex subunit 1-like protein 1target
MenadioneXanthine dehydrogenase/oxidaseenzyme
MenadioneAldehyde oxidaseenzyme
MenadioneMethylenetetrahydrofolate reductase (NADPH)enzyme
MenadioneCytochrome P450 1A1enzyme
MenadioneOsteocalcintarget
MenadioneCytochrome P450 1A2enzyme
MenadioneCytochrome P450 2A6enzyme
MenadioneCytochrome P450 1B1enzyme
MenadioneCytochrome P450 2B6enzyme
MenadioneCytochrome P450 2C8enzyme
MenadioneCytochrome P450 2C9enzyme
MenadioneCytochrome P450 2C19enzyme
MenadioneCytochrome P450 2D6enzyme
MenadioneCytochrome P450 2E1enzyme
MenadioneCytochrome P450 3A4enzyme
MenadioneCytochrome P450 3A5enzyme
MenadioneCytochrome P450 3A7enzyme
MenadioneAldehyde oxidasetarget
AlitretinoinRetinoic acid receptor alphatarget
AlitretinoinRetinoic acid receptor RXR-betatarget
AlitretinoinRetinoic acid receptor gammatarget
AlitretinoinRetinoic acid receptor betatarget
AlitretinoinRetinoic acid receptor RXR-gammatarget
AlitretinoinRetinoic acid receptor RXR-alphatarget
AlitretinoinCellular retinoic acid-binding protein 2carrier
AlitretinoinCellular retinoic acid-binding protein 1carrier
AlitretinoinATP-dependent translocase ABCB1transporter
AlitretinoinInsulin-like growth factor-binding protein 3target
AlitretinoinPregnancy-specific beta-1-glycoprotein 5target
AlitretinoinCytochrome P450 26C1target
TretinoinRetinoic acid receptor gammatarget
TretinoinRetinoic acid receptor RXR-betatarget
TretinoinAldehyde dehydrogenase 1A1target
TretinoinRetinoic acid-induced protein 3target
TretinoinRetinoic acid receptor RXR-gammatarget
TretinoinRetinal dehydrogenase 2target
TretinoinRetinoic acid receptor responder protein 1target
TretinoinCytochrome P450 2C8enzyme
TretinoinCellular retinoic acid-binding protein 1transporter
TretinoinCellular retinoic acid-binding protein 2transporter
TretinoinCytochrome P450 2B6enzyme
TretinoinCytochrome P450 3A4enzyme
TretinoinCytochrome P450 3A5enzyme
TretinoinCytochrome P450 2A6enzyme
TretinoinCytochrome P450 3A7enzyme
TretinoinCytochrome P450 2C18enzyme
TretinoinCytochrome P450 2C9enzyme
TretinoinCytochrome P450 4A11enzyme
TretinoinCytochrome P450 1A1enzyme
TretinoinRetinoic acid receptor alphatarget
TretinoinRetinoic acid receptor betatarget
TretinoinLipocalin-1target
TretinoinOdorant-binding protein 2atarget
TretinoinRetinol-binding protein 4target
TretinoinAlbumincarrier
Tretinoin[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 4, mitochondrialtarget
TretinoinRetinoic acid receptor RXR-alphatarget
TretinoinCarcinoembryonic antigentarget
TretinoinUDP-glucuronosyltransferase 2B7enzyme
TretinoinCytochrome P450 2E1enzyme
TretinoinCytochrome P450 26A1enzyme
TretinoinCellular retinoic acid-binding protein 1target
PaclitaxelApoptosis regulator Bcl-2target
PaclitaxelTubulin beta-1 chaintarget
PaclitaxelCytochrome P450 2C8enzyme
PaclitaxelCytochrome P450 3A4enzyme
PaclitaxelCytochrome P450 3A5enzyme
PaclitaxelCytochrome P450 3A7enzyme
PaclitaxelBile salt export pumptransporter
PaclitaxelATP-dependent translocase ABCB1transporter
PaclitaxelMultidrug resistance-associated protein 1transporter
PaclitaxelATP-binding cassette sub-family C member 10transporter
PaclitaxelAromataseenzyme
PaclitaxelCytochrome P450 1B1enzyme
PaclitaxelSolute carrier organic anion transporter family member 1B3transporter
PaclitaxelNuclear receptor subfamily 1 group I member 2target
PaclitaxelMicrotubule-associated protein 4target
PaclitaxelMicrotubule-associated protein 2target
PaclitaxelMicrotubule-associated protein tautarget
PaclitaxelATP-binding cassette sub-family C member 2transporter
DocetaxelApoptosis regulator Bcl-2target
DocetaxelTubulin beta-1 chaintarget
DocetaxelCytochrome P450 3A4enzyme
DocetaxelCytochrome P450 3A5enzyme
DocetaxelCytochrome P450 3A7enzyme
DocetaxelATP-dependent translocase ABCB1transporter
DocetaxelATP-binding cassette sub-family C member 10transporter
DocetaxelCytochrome P450 1B1enzyme
DocetaxelMicrotubule-associated protein 2target
DocetaxelMicrotubule-associated protein 4target
DocetaxelMicrotubule-associated protein tautarget
DocetaxelSolute carrier organic anion transporter family member 1B3transporter
DocetaxelSolute carrier family 22 member 7transporter
DocetaxelBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
DocetaxelATP-binding cassette sub-family C member 2transporter
DocetaxelMultidrug resistance-associated protein 1transporter
DocetaxelNuclear receptor subfamily 1 group I member 2target
CarboxyatractylosideADP/ATP translocase 1target
N-EthylretinamideRetinol-binding protein 4carrier
EcabetNADPH oxidase organizer 1target
EcabetUrease subunit alphatarget
Paclitaxel docosahexaenoic acidApoptosis regulator Bcl-2target
Ginkgolide AGlycine receptor subunit alpha-1target
Ginkgolide AGlycine receptor subunit alpha-2target
Ginkgolide AGlycine receptor subunit alpha-3target
Ginkgolide AGlycine receptor subunit betatarget
CabazitaxelCytochrome P450 3A4enzyme
CabazitaxelCytochrome P450 3A5enzyme
CabazitaxelCytochrome P450 2C8enzyme
CabazitaxelATP-dependent translocase ABCB1transporter
CabazitaxelBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
CabazitaxelTubulin beta-1 chaintarget
CabazitaxelSolute carrier organic anion transporter family member 1B1transporter
CabazitaxelSolute carrier organic anion transporter family member 1B3transporter
CabazitaxelAlbumincarrier
CabazitaxelLow-density lipoprotein receptorcarrier
CabazitaxelVery low-density lipoprotein receptorcarrier
CabazitaxelGlycosylphosphatidylinositol-anchored high density lipoprotein-binding protein 1carrier
Gibberellic acidArylacetamide deacetylase-like 2target
Gibberellin A4Arylacetamide deacetylase-like 2target
OrtataxelTumor necrosis factortarget
MenatetrenoneCruzipaintarget
Salvinorin AMu-type opioid receptortarget
Salvinorin ADelta-type opioid receptortarget
Salvinorin AKappa-type opioid receptortarget
MilataxelTubulin beta-1 chaintarget
MilataxelTubulin beta chaintarget
Phorbol 12-myristate 13-acetate diesterTransient receptor potential cation channel subfamily V member 4target
Phorbol 12-myristate 13-acetate diesterG protein-activated inward rectifier potassium channel 4target
AphidicolinDNA polymerase catalytic subunittarget