Cytochrome P-450 CYP2E1 Substrates with a Narrow Therapeutic Index

Name
Cytochrome P-450 CYP2E1 Substrates with a Narrow Therapeutic Index
Accession Number
DBCAT004032
Description

Not Available

Drugs
DrugDrug Description
QuinidineA medication used to restore normal sinus rhythm, treat atrial fibrillation and flutter, and treat ventricular arrhythmias.
DacarbazineAn antineoplastic agent used to treat malignant melanoma and Hodgkin's disease.
TrabectedinAn alkylating agent approved for the treatment of unresectable or metastatic soft tissue sarcoma (liposarcoma or leiomyosarcoma).
EtoposideA podophyllotoxin derivative used to treat testicular and small cell lung tumors.
TegafurAn antineoplastic agent used in combination with other anticancer medications to treat advanced gastric and colorectal cancers.
TamoxifenA selective estrogen receptor modulator used to treat estrogen receptor positive breast cancer, reduce the risk of invasive breast cancer following surgery, or reduce the risk of breast cancer in high risk women.
MitoxantroneA chemotherapeutic agent used for the treatment of secondary progressive, progressive relapsing, or worsening relapsing-remitting multiple sclerosis.
TheophyllineA xanthine used to manage the symptoms of asthma, COPD, and other lung conditions caused by reversible airflow obstruction.
AminophyllineA bronchodilator consisting of theophylline that is used for the treatment of bronchospasm due to asthma, emphysema and chronic bronchitis.
PhenobarbitalA long-lasting barbiturate and anticonvulsant used in the treatment of all types of seizures, except for absent seizures.
DalfampridineA potassium channel blocker used for the improvement of motor function in patients with multiple sclerosis (MS).
PhenytoinAn anticonvulsant drug used in the prophylaxis and control of various types of seizures.
Drugs & Drug Targets
DrugTargetType
QuinidineSodium channel protein type 5 subunit alphatarget
QuinidineAlpha-1-acid glycoprotein 1carrier
QuinidineVoltage-gated inwardly rectifying potassium channel KCNH2target
QuinidinePotassium channel subfamily K member 1target
QuinidinePotassium channel subfamily K member 6target
QuinidineCytochrome P450 1A2enzyme
QuinidineCytochrome P450 2E1enzyme
QuinidineCytochrome P450 1A1enzyme
QuinidineCytochrome P450 2D6enzyme
QuinidineCytochrome P450 3A4enzyme
QuinidineCytochrome P450 3A7enzyme
QuinidineSolute carrier family 22 member 2transporter
QuinidineSolute carrier family 22 member 1transporter
QuinidineOrganic cation/carnitine transporter 2transporter
QuinidineATP-dependent translocase ABCB1transporter
QuinidineSolute carrier organic anion transporter family member 1A2transporter
QuinidineOrganic anion transporter 3transporter
QuinidineATP-binding cassette sub-family C member 2transporter
QuinidineSolute carrier family 22 member 4transporter
QuinidineSolute carrier organic anion transporter family member 1B1transporter
QuinidineCytochrome P450 2B6enzyme
QuinidineCytochrome P450 2C9enzyme
QuinidineAlpha-1A adrenergic receptortarget
QuinidineAlpha-1B adrenergic receptortarget
QuinidineAlpha-1D adrenergic receptortarget
QuinidineBile salt export pumptransporter
QuinidineCytochrome P450 2C8enzyme
QuinidineAlbumincarrier
DacarbazineDNA polymerase alpha subunit Btarget
DacarbazineCytochrome P450 1A1enzyme
DacarbazineCytochrome P450 1A2enzyme
DacarbazineCytochrome P450 2E1enzyme
Dacarbazine6-phosphogluconate dehydrogenase, decarboxylatingtarget
DacarbazineDNAtarget
TrabectedinCytochrome P450 3A4enzyme
TrabectedinCytochrome P450 2C9enzyme
TrabectedinCytochrome P450 2D6enzyme
TrabectedinCytochrome P450 2E1enzyme
TrabectedinCytochrome P450 2C19enzyme
TrabectedinDNAtarget
TrabectedinProstaglandin G/H synthase 1enzyme
EtoposideDNA topoisomerase 2-alphatarget
EtoposideCytochrome P450 3A4enzyme
EtoposideATP-binding cassette sub-family C member 3transporter
EtoposideATP-binding cassette sub-family C member 6transporter
EtoposideATP-dependent translocase ABCB1transporter
EtoposideMultidrug resistance-associated protein 1transporter
EtoposideATP-binding cassette sub-family C member 10transporter
EtoposideATP-binding cassette sub-family C member 2transporter
EtoposideBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
EtoposideCytochrome P450 1A2enzyme
EtoposideCytochrome P450 2E1enzyme
EtoposideCytochrome P450 3A5enzyme
EtoposideUDP-glucuronosyltransferase 1A1enzyme
EtoposideDNA topoisomerase 2-betatarget
EtoposideGlutathione S-transferase theta-1enzyme
EtoposideGlutathione S-transferase Penzyme
EtoposideProstaglandin G/H synthase 2enzyme
EtoposideProstaglandin G/H synthase 1enzyme
TegafurCytochrome P450 2A6enzyme
TegafurThymidylate synthasetarget
TegafurCytochrome P450 1A2enzyme
TegafurCytochrome P450 2C8enzyme
TegafurCytochrome P450 2E1enzyme
TegafurCytochrome P450 3A5enzyme
TegafurThyroxine-binding globulincarrier
TamoxifenEstrogen receptortarget
TamoxifenEstrogen receptor betatarget
TamoxifenCytochrome P450 2C9enzyme
TamoxifenCytochrome P450 3A4enzyme
TamoxifenCytochrome P450 2D6enzyme
TamoxifenCytochrome P450 2C8enzyme
TamoxifenCytochrome P450 2B6enzyme
TamoxifenLiver carboxylesterase 1enzyme
TamoxifenCytochrome P450 3A5enzyme
TamoxifenCytochrome P450 1A1enzyme
TamoxifenCytochrome P450 1B1enzyme
TamoxifenCytochrome P450 2C19enzyme
TamoxifenFlavin-containing monooxygenase 1enzyme
TamoxifenFlavin-containing monooxygenase 3enzyme
TamoxifenCytochrome P450 3A7enzyme
TamoxifenATP-dependent translocase ABCB1transporter
TamoxifenBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
TamoxifenAromataseenzyme
TamoxifenCytochrome P450 2A6enzyme
TamoxifenCytochrome P450 2E1enzyme
TamoxifenUDP-glucuronosyltransferase 1A10enzyme
TamoxifenSulfotransferase 1A1enzyme
TamoxifenATP-binding cassette sub-family C member 2transporter
Tamoxifen3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerasetarget
TamoxifenProtein kinase Ctarget
TamoxifenAndrogen receptortarget
TamoxifenVoltage-gated inwardly rectifying potassium channel KCNH2target
TamoxifenNuclear receptor subfamily 1 group I member 2target
TamoxifenEstrogen-related receptor gammatarget
TamoxifenSex hormone-binding globulintarget
TamoxifenBile salt export pumptransporter
TamoxifenThyroxine-binding globulincarrier
TamoxifenSulfotransferase 2A1enzyme
TamoxifenCytochrome P450 1A2enzyme
TamoxifenUDP-glucuronosyltransferase 2B7enzyme
TamoxifenUDP-glucuronosyltransferase 2B17enzyme
TamoxifenSulfotransferase 1E1enzyme
TamoxifenPhospholipid-transporting ATPase ABCA1transporter
TamoxifenMitogen-activated protein kinase 8target
TamoxifenAlbumincarrier
MitoxantroneDNA topoisomerase 2-alphatarget
MitoxantroneCytochrome P450 2E1enzyme
MitoxantroneATP-dependent translocase ABCB1transporter
MitoxantroneMultidrug resistance-associated protein 1transporter
MitoxantroneBroad substrate specificity ATP-binding cassette transporter ABCG2transporter
MitoxantroneDNAtarget
MitoxantroneCytochrome P450 1B1enzyme
MitoxantroneCytochrome P450 3A4enzyme
MitoxantroneDNA topoisomerase 2-betatarget
TheophyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
Theophylline3',5'-cyclic-AMP phosphodiesterase 4Btarget
TheophyllineAdenosine receptor A2btarget
Theophylline3',5'-cyclic-AMP phosphodiesterase 4Atarget
TheophyllinecGMP-specific 3',5'-cyclic phosphodiesterasetarget
TheophyllineAdenosine receptor A1target
TheophyllineAdenosine receptor A2atarget
TheophyllineCytochrome P450 1A2enzyme
TheophyllineAdenosine deaminaseenzyme
TheophyllineCytochrome P450 2E1enzyme
TheophyllineCytochrome P450 3A4enzyme
TheophyllineSolute carrier family 22 member 7transporter
TheophyllineCytochrome P450 1A1enzyme
TheophyllineCytochrome P450 1B1enzyme
TheophyllineCytochrome P450 2D6enzyme
TheophyllineHistone deacetylase 2target
TheophyllineCopine-1target
TheophyllineMinor histocompatibility antigen H13target
TheophyllineBOS complex subunit NOMO1target
TheophyllinePoly [ADP-ribose] polymerase 1target
TheophyllineProtein RIC-3target
TheophyllineTubulin monoglycylase TTLL3target
Theophylline5'-nucleotidasetarget
AminophyllinecGMP-inhibited 3',5'-cyclic phosphodiesterase 3Atarget
AminophyllineAdenosine receptor A3target
AminophyllineAdenosine receptor A1target
AminophyllineCytochrome P450 1A2enzyme
AminophyllineCytochrome P450 2E1enzyme
AminophyllineCytochrome P450 3A4enzyme
AminophyllineHistone deacetylase 2target
PhenobarbitalGamma-aminobutyric acid receptor subunit alpha-1target
PhenobarbitalCytochrome P450 2C19enzyme
PhenobarbitalCytochrome P450 2C9enzyme
PhenobarbitalCytochrome P450 2B6enzyme
PhenobarbitalCytochrome P450 2C8enzyme
PhenobarbitalCytochrome P450 1A2enzyme
PhenobarbitalCytochrome P450 3A4enzyme
PhenobarbitalATP-binding cassette sub-family C member 3transporter
PhenobarbitalBile salt export pumptransporter
PhenobarbitalATP-dependent translocase ABCB1transporter
PhenobarbitalMultidrug resistance-associated protein 1transporter
PhenobarbitalSolute carrier organic anion transporter family member 2A1transporter
PhenobarbitalATP-binding cassette sub-family C member 2transporter
PhenobarbitalNeuronal acetylcholine receptor subunit alpha-4target
PhenobarbitalNeuronal acetylcholine receptor subunit alpha-7target
PhenobarbitalGlutamate receptor 2target
PhenobarbitalGlutamate receptor ionotropic, kainate 2target
PhenobarbitalCytochrome P450 2A6enzyme
PhenobarbitalCytochrome P450 2E1enzyme
PhenobarbitalCytochrome P450 3A5enzyme
PhenobarbitalCytochrome P450 1A1enzyme
PhenobarbitalCytochrome P450 2C18enzyme
PhenobarbitalCytochrome P450 3A7enzyme
PhenobarbitalCytochrome P450 4B1enzyme
PhenobarbitalNMDA receptortarget
PhenobarbitalNuclear receptor subfamily 1 group I member 2target
PhenobarbitalUDP-glucuronosyltransferase 1A1enzyme
PhenobarbitalUDP-glucuronosyltransferase 2B7enzyme
DalfampridineCytochrome P450 2E1enzyme
DalfampridineA-type voltage-gated potassium channel KCND2target
DalfampridineA-type voltage-gated potassium channel KCND3target
DalfampridinePotassium voltage-gated channel subfamily A member 1target
DalfampridinePotassium voltage-gated channel subfamily A member 4target
DalfampridinePotassium voltage-gated channel subfamily A member 2target
DalfampridinePotassium voltage-gated channel subfamily A member 3target
DalfampridinePotassium voltage-gated channel subfamily A member 5target
DalfampridinePotassium voltage-gated channel subfamily A member 6target
DalfampridinePotassium voltage-gated channel subfamily A member 7target
DalfampridinePotassium voltage-gated channel subfamily A member 10target
DalfampridinePotassium voltage-gated channel subfamily B member 1target
DalfampridinePotassium voltage-gated channel subfamily B member 2target
DalfampridineVoltage-gated potassium channel KCNC1target
DalfampridineVoltage-gated potassium channel KCNC2target
DalfampridineVoltage-gated potassium channel KCNC3target
DalfampridineA-type voltage-gated potassium channel KCND1target
DalfampridineSolute carrier family 22 member 2transporter
PhenytoinSodium channel protein type 5 subunit alphatarget
PhenytoinSodium channel protein type 1 subunit alphatarget
PhenytoinCytochrome P450 2C8enzyme
PhenytoinCytochrome P450 2C19enzyme
PhenytoinCytochrome P450 2C9enzyme
PhenytoinCytochrome P450 2B6enzyme
PhenytoinCytochrome P450 3A5enzyme
PhenytoinAlbumincarrier
PhenytoinCytochrome P450 3A4enzyme
PhenytoinSolute carrier organic anion transporter family member 1C1transporter
PhenytoinATP-dependent translocase ABCB1transporter
PhenytoinATP-binding cassette sub-family C member 2transporter
PhenytoinCytochrome P450 11B1, mitochondrialenzyme
PhenytoinCytochrome P450 3A7enzyme
PhenytoinNuclear receptor subfamily 1 group I member 2target
PhenytoinSodium channel regulatory subunit beta-1target
PhenytoinSodium channel protein type 3 subunit alphatarget
PhenytoinUDP-glucuronosyltransferase 1A1enzyme
PhenytoinUDP-glucuronosyltransferase 1-6enzyme
PhenytoinUDP-glucuronosyltransferase 1A9enzyme
PhenytoinThyroxine-binding globulincarrier
PhenytoinVoltage-gated inwardly rectifying potassium channel KCNH2target
PhenytoinVoltage-dependent L-type calcium channeltarget
PhenytoinSodium channel protein type 2 subunit alphatarget
PhenytoinSodium channel protein type 8 subunit alphatarget
PhenytoinGABA(A) Receptortarget
PhenytoinCytochrome P450 1A2enzyme
PhenytoinCytochrome P450 2A6enzyme
PhenytoinCytochrome P450 2D6enzyme
PhenytoinCytochrome P450 2E1enzyme
PhenytoinEpoxide hydrolase 1enzyme
PhenytoinUDP-glucuronosyltransferase 1A4enzyme
PhenytoinCatechol O-methyltransferaseenzyme
PhenytoinNAD(P)H dehydrogenase [quinone] 1enzyme
PhenytoinCytochrome P450 2C18enzyme